A facile synthesis of substituted pyridines and pyrazolo[3,4-b]pyridines

被引：7
|
作者：
Kidwai, M [1 ]
Thakur, R [1 ]
Saxena, S [1 ]
机构：
[1] Univ Delhi, Dept Chem, Delhi 110007, India
来源：
JOURNAL OF HETEROCYCLIC CHEMISTRY | 2005年 / 42卷 / 06期
关键词：
D O I：
10.1002/jhet.5570420622
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A facile, solvent free, ecoffiendly approach for the synthesis of 2-amino-3(ethylcarboxy)-4,6-disubstituted pyridine 4 and pyrazolo[3,4-b]pyridines 6 is herein described employing neat reaction conditions under microwave irradiation. This solventless methodology is environmentally benign as it completely eliminates the use of solvent from the reaction procedure. The observed reaction rate enhancement and high yield of products are due to the neat reaction conditions coupled with microwaves (MWs).
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收藏
页码：1181 / 1183
页数：3
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