HIV-1 Integrase Strand Transfer Inhibitors

被引：1
|
作者：
Johns, Brian A. [1 ]
机构：
[1] GlaxoSmithKline, Res Triangle Pk, NC 27709 USA
来源：
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 45 | 2010年 / 45卷
关键词：
TREATMENT-NAIVE; ANTIRETROVIRAL ACTIVITY; ANTIVIRAL ACTIVITY; PART; RALTEGRAVIR; RESISTANCE; PHARMACOKINETICS; ELVITEGRAVIR; SAFETY; POTENT;
D O I：
10.1016/S0065-7743(10)45016-2
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：263 / +
页数：15
相关论文
共 50 条
  • [1] Targeting HIV-1 integrase with strand transfer inhibitors
    Li, Yang
    Xuan, Shouyi
    Feng, Yue
    Yan, Aixia
    [J]. DRUG DISCOVERY TODAY, 2015, 20 (04) : 435 - 449
  • [2] HIV-1 Integrase Strand Transfer Inhibitors and Neurodevelopment
    Foster, Emma G.
    Gendelman, Howard E.
    Bade, Aditya N.
    [J]. PHARMACEUTICALS, 2022, 15 (12)
  • [3] Chromone and chromanone derivatives as strand transfer inhibitors of HIV-1 integrase
    Park, Jang Hyun
    Lee, Seung Uk
    Kim, Sang Hoon
    Shin, Seo Yeong
    Lee, Jae Yeol
    Shin, Cha-Gyun
    Yoo, Kyung Ho
    Lee, Yong Sup
    [J]. ARCHIVES OF PHARMACAL RESEARCH, 2008, 31 (01) : 1 - 5
  • [4] Ruthenium arene complexes as HIV-1 integrase strand transfer inhibitors
    Carcelli, Mauro
    Bacchi, Alessia
    Pelagatti, Paolo
    Rispoli, Gabriele
    Rogolino, Dominga
    Sanchez, Tino W.
    Sechi, Mario
    Neamati, Nouri
    [J]. JOURNAL OF INORGANIC BIOCHEMISTRY, 2013, 118 : 74 - 82
  • [5] Chromone and chromanone derivatives as strand transfer inhibitors of HIV-1 integrase
    Jang Hyun Park
    Seung Uk Lee
    Sang Hoon Kim
    Seo Yeong Shin
    Jae Yeol Lee
    Cha-Gyun Shin
    Kyung Ho Yoo
    Yong Sup Lee
    [J]. Archives of Pharmacal Research, 2008, 31 : 1 - 5
  • [6] Inhibition of matrix metalloproteinases by HIV-1 integrase strand transfer inhibitors
    Foster, Emma G. G.
    Palermo, Nicholas Y. Y.
    Liu, Yutong
    Edagwa, Benson
    Gendelman, Howard E. E.
    Bade, Aditya N. N.
    [J]. FRONTIERS IN TOXICOLOGY, 2023, 5
  • [7] Comparative Clinical Pharmacokinetics and Pharmacodynamics of HIV-1 Integrase Strand Transfer Inhibitors
    Podany, Anthony T.
    Scarsi, Kimberly K.
    Fletcher, Courtney V.
    [J]. CLINICAL PHARMACOKINETICS, 2017, 56 (01) : 25 - 40
  • [8] Comparative Clinical Pharmacokinetics and Pharmacodynamics of HIV-1 Integrase Strand Transfer Inhibitors
    Anthony T. Podany
    Kimberly K. Scarsi
    Courtney V. Fletcher
    [J]. Clinical Pharmacokinetics, 2017, 56 : 25 - 40
  • [9] Investigating the Role of Metal Chelation in HIV-1 Integrase Strand Transfer Inhibitors
    Bacchi, Alessia
    Carcelli, Mauro
    Compari, Carlotta
    Fisicaro, Emilia
    Pala, Nicolino
    Rispoli, Gabriele
    Rogolino, Dominga
    Sanchez, Tino W.
    Sechi, Mario
    Sinisi, Valentina
    Neamati, Nouri
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2011, 54 (24) : 8407 - 8420
  • [10] Biochemical analysis of HIV-1 integrase variants resistant to strand transfer inhibitors
    Dicker, Ira B.
    Terry, Brian
    Lin, Zeyu
    Li, Zhufang
    Bollini, Sagarika
    Samanta, Himadri K.
    Gali, Volodymyr
    Walker, Michael A.
    Krystal, Mark R.
    [J]. JOURNAL OF BIOLOGICAL CHEMISTRY, 2008, 283 (35) : 23599 - 23609
12345