Synthesis and biological evaluation of alkenyldiarylmethane HIV-1 non-nucleoside reverse transcriptase inhibitors that possess increased hydrolytic stability

被引:0
|
作者
Cullen, Matthew D. [1 ]
De Clercq, Erik [2 ]
Pannecouque, Christophe
Hartman, Tracy L. [3 ]
Buckheit, Robert W., Jr. [3 ]
Deng, Bo Liang [5 ]
Cushman, Mark [1 ,4 ]
机构
[1] Purdue Univ, Dept Med Chem & Mol Pharmacol, W Lafayette, IN 47907 USA
[2] Katholieke Univ Leuven, Rega Inst Med Res, Johnson & Johnson Pharmaceut Res & Dev, B-3000 Louvain, Belgium
[3] Imquest Biosci Inc, Antiinfect Res, Frederick, MD 21704 USA
[4] Purdue Univ, Purdue Canc Ctr, W Lafayette, IN 47907 USA
[5] Nektar Therapeut, Huntsville, AL 35806 USA
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
72-MEDI
引用
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页码:666 / 666
页数:1
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