Synthesis of imidazo[1,2-a]pyridines: a decade update

被引：557
|
作者：
Bagdi, Avik Kumar [1 ]
Santra, Sougata [1 ]
Monir, Kamarul [1 ]
Hajra, Alakananda [1 ]
机构：
[1] Visva Bharati Cent Univ, Dept Chem, Santini Ketan 731235, W Bengal, India
来源：
CHEMICAL COMMUNICATIONS | 2015年 / 51卷 / 09期
关键词：
ONE-POT SYNTHESIS; INTRAMOLECULAR PROTON-TRANSFER; 3-COMPONENT REACTION; MULTICOMPONENT REACTION; FACILE SYNTHESIS; 2-AMINOPYRIDINES; DERIVATIVES; CYCLIZATION; CATALYST; ACCESS;
D O I：
10.1039/c4cc08495k
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Imidazopyridine is one of the important fused bicyclic 5-6 heterocycles and it is recognized as a "drug prejudice" scaffold due to its wide range of applications in medicinal chemistry. This moiety is also useful in material science because of its structural character. Synthesis of this moiety from the easily available chemicals is desirable due to its tremendous use in the various branches of chemistry. Here we report a review on the synthesis of this scaffold employing different strategies such as condensation, multicomponent reactions, oxidative coupling, tandem reactions, aminooxygenation, and hydroamination reactions.
引用
收藏
页码：1555 / 1575
页数：21
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