Affinity of dopamine for the D3 and D2 high receptors in the human brain in vivo

被引:0
|
作者
Rabiner, Eugenii [1 ]
Shotbolt, Paul [1 ]
Tziortzi, Andri [1 ]
Searle, Graham [1 ]
Laruelle, Marc [2 ]
Gunn, Roger [1 ]
机构
[1] GlaxoSmithKline, Clin Imaging Ctr, London, England
[2] GlaxoSmithKline, Neurosci CEDD, Harlow, Essex, England
关键词
D O I
暂无
中图分类号
R8 [特种医学]; R445 [影像诊断学];
学科分类号
1002 ; 100207 ; 1009 ;
摘要
497
引用
收藏
页数:2
相关论文
共 50 条
  • [1] (-)S amisulpride binds with high affinity to cloned dopamine D3 and D2 receptors
    Castelli, MP
    Mocci, I
    Sanna, AM
    Gessa, GL
    Pani, L
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 2001, 432 (2-3) : 143 - 147
  • [2] Regulation of Akt signaling by D2 and D3 dopamine receptors in vivo
    Beaulieu, Jean-Martin
    Tirotta, Emanuele
    Sotnikova, Tatyana D.
    Masri, Bernard
    Salahpour, Ali
    Gainetdinov, Raul R.
    Borrelli, Emiliana
    Caron, Marc G.
    [J]. JOURNAL OF NEUROSCIENCE, 2007, 27 (04): : 881 - 885
  • [3] DISTRIBUTION OF DOPAMINE D2, D3 AND D4 RECEPTORS IN HUMAN POSTMORTEM BRAIN SECTIONS
    LAHTI, RA
    CONLEY, R
    GRUBOWSKI, L
    TAMMINGA, CA
    [J]. SCHIZOPHRENIA RESEARCH, 1995, 15 (1-2) : 63 - 63
  • [4] Dopamine D2/D3 receptors in human retinal precursor cells
    Chu, J
    Xu, K
    Chu, TC
    [J]. FASEB JOURNAL, 2003, 17 (04): : A633 - A633
  • [5] In vitro pharmacology of antipsychotics at human dopamine D2 and D3 receptors
    Tadori, Yoshihiro
    Kobayashi, Hiroyuki
    [J]. JOURNAL OF PHARMACOLOGICAL SCIENCES, 2014, 124 : 70P - 70P
  • [6] Affinity and selectivity determinants of bitropic ligands targeting D2 and D3 dopamine receptors
    Hayatshahi, Hamed
    Luedtke, Robert
    Liu, Jin
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2019, 257
  • [7] Fluorescent ligands for dopamine D2/D3 receptors
    Anni Allikalt
    Nirupam Purkayastha
    Khajidmaa Flad
    Maximilian F. Schmidt
    Alina Tabor
    Peter Gmeiner
    Harald Hübner
    Dorothee Weikert
    [J]. Scientific Reports, 10
  • [8] Fluorescent ligands for dopamine D2/D3 receptors
    Allikalt, Anni
    Purkayastha, Nirupam
    Flad, Khajidmaa
    Schmidt, Maximilian F.
    Tabor, Alina
    Gmeiner, Peter
    Huebner, Harald
    Weikert, Dorothee
    [J]. SCIENTIFIC REPORTS, 2020, 10 (01)
  • [9] Functional potencies of dopamine agonists and antagonists at human dopamine D2 and D3 receptors
    Tadori, Yoshihiro
    Forbes, Robert A.
    McQuade, Robert D.
    Kikuchi, Tetsuro
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 2011, 666 (1-3) : 43 - 52
  • [10] In vitro characterisation of the high affinity D2/D3 dopamine agonist (+)PhNO
    Parker, Christine
    Clarke, K.
    Gee, A. D.
    Gee, A.
    Rabiner, E.
    [J]. NEUROIMAGE, 2006, 31 : T29 - T29