Novel radioiodinated P-glycoprotein inhibitors for SPECT imaging applications

被引:0
|
作者
Marina, Sagnou [1 ]
Dimitra, Benaki [1 ]
Antonis, Kostopoulos [2 ]
David, Dickens [3 ]
Charalambos, Triantis [2 ]
Stavros, Xanthopoulos [2 ]
Sotiris, Kakabakos [2 ]
Maria, Pelecanou [1 ]
Varvarigou, Alexandra D. [2 ]
机构
[1] Natl Ctr Sci Res Demokritos, Inst Biol, Athens, Greece
[2] Natl Ctr Sci Res Demokritos, Inst Radioisotopes Radiodiagnost Prod, Athens, Greece
[3] Univ Liverpool, Dept Pharmacol, Liverpool L69 3BX, Merseyside, England
来源
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2011年 / 54卷
关键词
D O I
暂无
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:S302 / S302
页数:1
相关论文
共 50 条
  • [1] Dibenzocyclooctadiene lingnans: a class of novel inhibitors of P-glycoprotein
    Qiangrong Pan
    Qinghua Lu
    Kun Zhang
    Xun Hu
    Cancer Chemotherapy and Pharmacology, 2006, 58 : 99 - 106
  • [2] Dibenzocyclooctadiene lingnans: a class of novel inhibitors of P-glycoprotein
    Pan, QR
    Lu, QH
    Zhang, K
    Hu, X
    CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2006, 58 (01) : 99 - 106
  • [3] Integrated approach to indentify novel P-glycoprotein substrates and inhibitors
    Bahadduri, Praveen
    Chang, Cheng
    Ekins, Sean
    Swaan, Peter
    FASEB JOURNAL, 2007, 21 (06): : A1188 - A1188
  • [4] Identification of Novel Inhibitors of P-glycoprotein Mediated Multidrug Resistance
    Follit, Courtney A.
    McCormick, James W.
    Nanayakkara, Amila K.
    Wise, John G.
    Vogel, Pia D.
    FASEB JOURNAL, 2017, 31
  • [5] Original Vinca Derivatives: From P-Glycoprotein Substrates to P-Glycoprotein Inhibitors
    Gherbovet, Olga
    Alvarez, Maria Concepcion Garcia
    Bignon, Jerome
    Roussi, Fanny
    JOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (23) : 10774 - 10780
  • [6] Imaging the Function of P-Glycoprotein With Radiotracers: Pharmacokinetics and In Vivo Applications
    Kannan, P.
    John, C.
    Zoghbi, S. S.
    Halldin, C.
    Gottesman, M. M.
    Innis, R. B.
    Hall, M. D.
    CLINICAL PHARMACOLOGY & THERAPEUTICS, 2009, 86 (04) : 368 - 377
  • [7] Substrates, Inhibitors and Activators of P-glycoprotein: Candidates for Radiolabeling and Imaging Perspectives
    Colabufo, Nicola A.
    Berardi, Francesco
    Perrone, Maria Grazia
    Capparelli, Elena
    Cantore, Mariangela
    Inglese, Carmela
    Perrone, Roberto
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2010, 10 (17) : 1703 - 1714
  • [8] Characterization of P-Glycoprotein Inhibitors for Evaluating the Effect of P-Glycoprotein on the Intestinal Absorption of Drugs
    Kono, Yusuke
    Kawahara, Iichiro
    Shinozaki, Kohei
    Nomura, Ikuo
    Marutani, Honoka
    Yamamoto, Akira
    Fujita, Takuya
    PHARMACEUTICS, 2021, 13 (03)
  • [9] Novel in vitro transport method for screening the reversibility of P-glycoprotein inhibitors
    Netsomboon, Kesinee
    Laffleur, Flavia
    Suchaoin, Wongsakorn
    Bernkop-Schnurch, Andreas
    EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS, 2016, 100 : 9 - 14
  • [10] ERBB and P-glycoprotein inhibitors break resistance in relapsed neuroblastoma models through P-glycoprotein
    Roesch, Lisa
    Herter, Sonja
    Najafi, Sara
    Ridinger, Johannes
    Peterziel, Heike
    Cinatl, Jindrich
    Jones, David T. W.
    Michaelis, Martin
    Witt, Olaf
    Oehme, Ina
    MOLECULAR ONCOLOGY, 2023, 17 (01) : 37 - 58