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- [1] Identification of aurintricarboxylic acid as a potent allosteric antagonist of P2X1 and P2X3 receptorsNEUROPHARMACOLOGY, 2019, 158Obrecht, Astrid S.论文数: 0 引用数: 0 h-index: 0机构: Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, Germany Univ Hosp RWTH Aachen, Dept Plast Surg Hand & Burn Surg, Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanyUrban, Nicole论文数: 0 引用数: 0 h-index: 0机构: Univ Leipzig, Rudolf Boehm Inst Pharmacol & Toxicol, D-04107 Leipzig, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanySchaefer, Michael论文数: 0 引用数: 0 h-index: 0机构: Univ Leipzig, Rudolf Boehm Inst Pharmacol & Toxicol, D-04107 Leipzig, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanyRoese, Anni论文数: 0 引用数: 0 h-index: 0机构: Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanyKless, Achim论文数: 0 引用数: 0 h-index: 0机构: Grunenthal GmbH, Dept Translat Sci & Intelligence, Grunenthal Innovat, D-52078 Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanyMeents, Jannis E.论文数: 0 引用数: 0 h-index: 0机构: Rhein Westfal TH Aachen, Inst Physiol, D-52074 Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanyLampert, Angelika论文数: 0 引用数: 0 h-index: 0机构: Rhein Westfal TH Aachen, Inst Physiol, D-52074 Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanyAbdelrahman, Aliaa论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, PharmaCtr Bonn, Pharmaceut Inst, Pharmaceut Chem 1, D-53121 Bonn, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanyMueller, Christa E.论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, PharmaCtr Bonn, Pharmaceut Inst, Pharmaceut Chem 1, D-53121 Bonn, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanySchmalzing, Gunther论文数: 0 引用数: 0 h-index: 0机构: Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, GermanyHausmann, Ralf论文数: 0 引用数: 0 h-index: 0机构: Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, D-52074 Aachen, Germany
- [2] High-throughput screening of approved drugs and bioactive compounds identifies aurintricarboxylic acid as a nanomolar potent antagonist of the P2X3 receptorNAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2017, 390 : S42 - S42Obrecht, A.论文数: 0 引用数: 0 h-index: 0机构: Rhein Westfal TH Aachen, Mol Pharmacol, Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, Aachen, GermanyUrban, N.论文数: 0 引用数: 0 h-index: 0机构: Univ Leipzig, Rudolf Boehm Inst Pharmacol & Toxicol, Leipzig, Germany Rhein Westfal TH Aachen, Mol Pharmacol, Aachen, GermanySchaefer, M.论文数: 0 引用数: 0 h-index: 0机构: Univ Leipzig, Rudolf Boehm Inst Pharmacol & Toxicol, Leipzig, Germany Rhein Westfal TH Aachen, Mol Pharmacol, Aachen, GermanySchmalzing, G.论文数: 0 引用数: 0 h-index: 0机构: Rhein Westfal TH Aachen, Mol Pharmacol, Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, Aachen, GermanyHausmann, R.论文数: 0 引用数: 0 h-index: 0机构: Rhein Westfal TH Aachen, Mol Pharmacol, Aachen, Germany Rhein Westfal TH Aachen, Mol Pharmacol, Aachen, Germany
- [3] Druggable negative allosteric site of P2X3 receptorsPROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 115 (19) : 4939 - 4944Wang, Jin论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R China Shanghai Jiao Tong Univ, Sch Med, Inst Med Sci, Dept Pharmacol & Chem Biol, Shanghai 200025, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaWang, Yao论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R China Shanghai Jiao Tong Univ, Sch Med, Inst Med Sci, Dept Pharmacol & Chem Biol, Shanghai 200025, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaCui, Wen-Wen论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Med, Inst Med Sci, Dept Pharmacol & Chem Biol, Shanghai 200025, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaHuang, Yichen论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaYang, Yang论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Med, Inst Med Sci, Dept Pharmacol & Chem Biol, Shanghai 200025, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaLiu, Yan论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Med, Inst Med Sci, Dept Pharmacol & Chem Biol, Shanghai 200025, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaZhao, Wen-Shan论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Med, Inst Med Sci, Dept Pharmacol & Chem Biol, Shanghai 200025, Peoples R China Lanzhou Univ, Sch Basic Med Sci, Key Lab Preclin Study New Drugs Gansu Prov, Lanzhou 730000, Gansu, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaCheng, Xiao-Yang论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Med, Inst Med Sci, Dept Pharmacol & Chem Biol, Shanghai 200025, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaSun, Wang-Sheng论文数: 0 引用数: 0 h-index: 0机构: Lanzhou Univ, Sch Basic Med Sci, Key Lab Preclin Study New Drugs Gansu Prov, Lanzhou 730000, Gansu, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaCao, Peng论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Hosp Integrated Tradit Chinese & Western Med, Nanjing 210023, Jiangsu, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaZhu, Michael X.论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 200025, Peoples R China Univ Texas Hlth Sci Ctr Houston, McGovern Med Sch, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaWang, Rui论文数: 0 引用数: 0 h-index: 0机构: Lanzhou Univ, Sch Basic Med Sci, Key Lab Preclin Study New Drugs Gansu Prov, Lanzhou 730000, Gansu, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaHattori, Motoyuki论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R ChinaYu, Ye论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Med, Inst Med Sci, Dept Pharmacol & Chem Biol, Shanghai 200025, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 200025, Peoples R China Fudan Univ, Collaborat Innovat Ctr Genet & Dev, Sch Life Sci, Dept Physiol & Biophys,State Key Lab Genet Engn, Shanghai 200438, Peoples R China
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- [7] A-317491, a novel potent and selective nonnucleotide antagonist of P2X3 and P2X2/3 receptors, reduces chronic inflammatory and neuropathic pain in the ratPROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2002, 99 (26) : 17179 - 17184Jarvis, MF论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USABurgard, EC论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAMcGaraughty, S论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAHonore, P论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USALynch, K论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USABrennan, TJ论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USASubieta, A论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAvan Biesen, T论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USACartmell, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USABianchi, B论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USANiforatos, W论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAKage, K论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAYu, HX论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAMikusa, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAWismer, CT论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAZhu, CZ论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAChu, K论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USALee, CH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAStewart, AO论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAPolakowski, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USACox, BF论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAKowaluk, E论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAWilliams, M论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USASullivan, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USAFaltynek, C论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Neurosci Res, Abbott Pk, IL 60064 USA
- [8] Discovery of Potent Antiallodynic Agents for Neuropathic Pain Targeting P2X3 ReceptorsACS CHEMICAL NEUROSCIENCE, 2017, 8 (07): : 1465 - 1478Jung, Young-Hwan论文数: 0 引用数: 0 h-index: 0机构: Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South Korea论文数: 引用数: h-index:机构:Lin, Hai论文数: 0 引用数: 0 h-index: 0机构: Chonnam Natl Univ, Med Sch, Dept Anesthesiol & Pain Med, Gwangju 501757, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South KoreaCho, Joong-Heui论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn DGMIF, New Drug Dev Ctr NDDC, 80 Cheombok Ro, Daegu 41061, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South KoreaPark, Jin-Hee论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn DGMIF, New Drug Dev Ctr NDDC, 80 Cheombok Ro, Daegu 41061, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South KoreaLee, So-Deok论文数: 0 引用数: 0 h-index: 0机构: Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South KoreaBae, Jinsu论文数: 0 引用数: 0 h-index: 0机构: Gwangju Inst Sci & Technol GIST, Dept Biomed Sci & Engn, Gwangju 500712, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South KoreaKang, Koon Mook论文数: 0 引用数: 0 h-index: 0机构: Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South KoreaKim, Moon-Gyoon论文数: 0 引用数: 0 h-index: 0机构: Dankook Univ, Coll Pharm, Cheonan 330714, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South KoreaPae, Ae Nim论文数: 0 引用数: 0 h-index: 0机构: Korea Inst Sci & Technol, Convergence Res Ctr Diag Treatment & Care Syst De, POB 131, Seoul 130650, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South KoreaKo, Hyojin论文数: 0 引用数: 0 h-index: 0机构: Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South Korea论文数: 引用数: h-index:机构:Yoon, Myung Ha论文数: 0 引用数: 0 h-index: 0机构: Chonnam Natl Univ, Med Sch, Dept Anesthesiol & Pain Med, Gwangju 501757, South Korea Chonnam Natl Univ, Med Sch, Ctr Creat Biomed Scientists, Gwangju 501757, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South KoreaKim, Yong-Chul论文数: 0 引用数: 0 h-index: 0机构: Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South Korea Gwangju Inst Sci & Technol GIST, Dept Biomed Sci & Engn, Gwangju 500712, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju 500712, South Korea
- [9] A Single Amino Acid Mutation Turns a P2X3 Antagonist into an AgonistBIOPHYSICAL JOURNAL, 2009, 96 (03) : 485A - 485AWang, Jixin论文数: 0 引用数: 0 h-index: 0机构: Merck, MRL, Pain Res, West Point, PA USA Merck, MRL, Pain Res, West Point, PA USAMoore, Eric论文数: 0 引用数: 0 h-index: 0机构: Merck, MRL, Pain Res, West Point, PA USA Merck, MRL, Pain Res, West Point, PA USAKane, Stefanie论文数: 0 引用数: 0 h-index: 0机构: Merck, MRL, Pain Res, West Point, PA USA Merck, MRL, Pain Res, West Point, PA USASalvatore, Christopher论文数: 0 引用数: 0 h-index: 0机构: Merck, MRL, Pain Res, West Point, PA USA Merck, MRL, Pain Res, West Point, PA USACook, Sean论文数: 0 引用数: 0 h-index: 0机构: Merck, MRL, Pain Res, West Point, PA USA Merck, MRL, Pain Res, West Point, PA USA
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