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- [1] MEDI 346-Preparation of sEH inhibitors with improved drug-like propertiesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 233 : 858 - 858Kort, Michael E.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USADrizin, Irene论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAGregg, Robert J.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAScanio, Marc J. C.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAShi, Lei论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAGross, Michael F.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAAtkinson, Robert N.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAJohnson, Matthew S.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAPacofsky, Gregory F.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASecrest, Matthew E.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAThomas, James B.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USACarroll, William A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMarron, Brian E.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAChapman, Mark L.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAKrambis, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALiu, Dong论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAShieh, Char-Chang论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAZhang, XuFeng论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAHernandez, Gricelda论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMikusa, Joseph P.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAZhong, Chengmin论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAJoshi, Shailen论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAHonore, Prisca论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USARoeloffs, Rosemarie论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMarsh, Kennan C.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMurray, Bernard P.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALiu, Jinrong论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAWerness, Stephen论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAFaltynek, Connie R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAKrafte, Douglas S.论文数: 0 引用数: 0 h-index: 0机构: Icagen Inc, Durham, NC 27703 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAJarvis, Michael F.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA
- [2] Improved drug-like properties of therapeutic proteins by directed evolutionPROTEIN ENGINEERING DESIGN & SELECTION, 2012, 25 (10): : 631 - 638Buchanan, Andrew论文数: 0 引用数: 0 h-index: 0机构: MedImmune Res, Cambridge CB21 6GH, England MedImmune Res, Cambridge CB21 6GH, EnglandFerraro, Franco论文数: 0 引用数: 0 h-index: 0机构: MedImmune Res, Cambridge CB21 6GH, England MedImmune Res, Cambridge CB21 6GH, EnglandRust, Steven论文数: 0 引用数: 0 h-index: 0机构: MedImmune Res, Cambridge CB21 6GH, England MedImmune Res, Cambridge CB21 6GH, EnglandSridharan, Sudharsan论文数: 0 引用数: 0 h-index: 0机构: MedImmune Res, Cambridge CB21 6GH, England MedImmune Res, Cambridge CB21 6GH, EnglandFranks, Ruth论文数: 0 引用数: 0 h-index: 0机构: MedImmune Res, Cambridge CB21 6GH, England MedImmune Res, Cambridge CB21 6GH, EnglandDean, Greg论文数: 0 引用数: 0 h-index: 0机构: MedImmune Res, Cambridge CB21 6GH, England MedImmune Res, Cambridge CB21 6GH, EnglandMcCourt, Matthew论文数: 0 引用数: 0 h-index: 0机构: MedImmune Res, Cambridge CB21 6GH, England MedImmune Res, Cambridge CB21 6GH, EnglandJermutus, Lutz论文数: 0 引用数: 0 h-index: 0机构: MedImmune Res, Cambridge CB21 6GH, England MedImmune Res, Cambridge CB21 6GH, EnglandMinter, Ralph论文数: 0 引用数: 0 h-index: 0机构: MedImmune Res, Cambridge CB21 6GH, England MedImmune Res, Cambridge CB21 6GH, England
- [3] Design and synthesis of chromone-based monoamine oxidase B inhibitors with improved drug-like propertiesEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 239论文数: 引用数: h-index:机构:Fernandes, Carlos论文数: 0 引用数: 0 h-index: 0机构: Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, Portugal Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalSalem, Hoda论文数: 0 引用数: 0 h-index: 0机构: Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, Portugal Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalMaia, Marta论文数: 0 引用数: 0 h-index: 0机构: Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, Portugal Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalTome, Claudia论文数: 0 引用数: 0 h-index: 0机构: Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, Portugal Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalBenfeito, Sofia论文数: 0 引用数: 0 h-index: 0机构: Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, Portugal Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalTeixeira, Jose论文数: 0 引用数: 0 h-index: 0机构: Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, Portugal Univ Coimbra, CNC Ctr Neurosci & Cell Biol, UC Biotech Bldg,Biocant Pk, P-3060197 Cantanhede, Portugal Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalOliveira, Paulo J.论文数: 0 引用数: 0 h-index: 0机构: Univ Coimbra, CNC Ctr Neurosci & Cell Biol, UC Biotech Bldg,Biocant Pk, P-3060197 Cantanhede, Portugal Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalUriarte, Eugenio论文数: 0 引用数: 0 h-index: 0机构: Univ Santiago de Compostela, Fac Pharm, Dept Organ Chem, Santiago De Compostela 15782, Spain Univ Autonoma Chile, Appl Chem Sci Inst, Santiago 7500912, Chile Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalOrtuso, Francesco论文数: 0 引用数: 0 h-index: 0机构: Univ Magna Grcecia Catanzaro, Dipartimento Sci Salute, Campus Salvatore Venuta,Viale Europa, I-88100 Catanzaro, Italy Univ Magna Grcecia Catanzaro, Net4Sci Srl, Acad Spinoff, Campus Salvatore Venuta,Viale Europa, I-88100 Catanzaro, Italy Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalAlcaro, Stefano论文数: 0 引用数: 0 h-index: 0机构: Univ Magna Grcecia Catanzaro, Dipartimento Sci Salute, Campus Salvatore Venuta,Viale Europa, I-88100 Catanzaro, Italy Univ Magna Grcecia Catanzaro, Net4Sci Srl, Acad Spinoff, Campus Salvatore Venuta,Viale Europa, I-88100 Catanzaro, Italy Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalBagetta, Donatella论文数: 0 引用数: 0 h-index: 0机构: Univ Magna Grcecia Catanzaro, Net4Sci Srl, Acad Spinoff, Campus Salvatore Venuta,Viale Europa, I-88100 Catanzaro, Italy Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalCagide, Fernando论文数: 0 引用数: 0 h-index: 0机构: Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, Portugal Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, PortugalBorges, Fernanda论文数: 0 引用数: 0 h-index: 0机构: Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, Portugal Univ Porto, Fac Sci, Dept Chem & Biochem, CIQUP IMS, P-4169007 Porto, Portugal
- [4] Synthesis and optimization of stapled DOCK peptides with improved drug-like propertiesARKIVOC, 2024, : 1 - 17Theppawong, Atiruj论文数: 0 引用数: 0 h-index: 0机构: Univ Ghent, Dept Organ & Macromol Chem, Krijgslaan 281 S4, B-9000 Ghent, Belgium Univ Ghent, Dept Organ & Macromol Chem, Krijgslaan 281 S4, B-9000 Ghent, BelgiumDe Geyter, Ewout论文数: 0 引用数: 0 h-index: 0机构: Univ Ghent, Dept Organ & Macromol Chem, Krijgslaan 281 S4, B-9000 Ghent, Belgium Univ Ghent, Dept Organ & Macromol Chem, Krijgslaan 281 S4, B-9000 Ghent, BelgiumMadder, Annemieke论文数: 0 引用数: 0 h-index: 0机构: Univ Ghent, Dept Organ & Macromol Chem, Krijgslaan 281 S4, B-9000 Ghent, Belgium Univ Ghent, Dept Organ & Macromol Chem, Krijgslaan 281 S4, B-9000 Ghent, Belgium
- [5] Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditionsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 246Papa, Alessandro论文数: 0 引用数: 0 h-index: 0机构: Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Cammarota, Mariarosaria论文数: 0 引用数: 0 h-index: 0机构: Univ Napoli Federico II, Dipartimento Neurosci & Sci Riprodutt Odontostomat, Div Farmacol, Via Pansini 5, I-80131 Naples, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, ItalyContri, Chiara论文数: 0 引用数: 0 h-index: 0机构: Univ Ferrara, Dipartimento Med Traslaz, Via Borsari 46, I-44121 Ferrara, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy论文数: 引用数: h-index:机构:Gemma, Sandra论文数: 0 引用数: 0 h-index: 0机构: Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy论文数: 引用数: h-index:机构:Lamponi, Stefania论文数: 0 引用数: 0 h-index: 0机构: Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, ItalyGorelli, Beatrice论文数: 0 引用数: 0 h-index: 0机构: Univ Siena, Dipartiment Sci Vita, Via Aldo Moro 2, I-53100 Siena, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Boscia, Francesca论文数: 0 引用数: 0 h-index: 0机构: Univ Napoli Federico II, Dipartimento Neurosci & Sci Riprodutt Odontostomat, Div Farmacol, Via Pansini 5, I-80131 Naples, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy论文数: 引用数: h-index:机构:Lodola, Alessio论文数: 0 引用数: 0 h-index: 0机构: Univ Parma, Dipartimento Sci Alimenti & Farmaco, Parco Area Sci 27-A, I-43124 Parma, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, ItalyButini, Stefania论文数: 0 引用数: 0 h-index: 0机构: Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, Via Aldo Moro 2, I-53100 Siena, Italy
- [6] Drug-like properties of tyrosine kinase inhibitors in ophthalmology: Formulation and topical availabilityINTERNATIONAL JOURNAL OF PHARMACEUTICS, 2024, 655论文数: 引用数: h-index:机构:Loftsson, Thorsteinn论文数: 0 引用数: 0 h-index: 0机构: Univ Iceland, Fac Pharmaceut Sci, Hofsvallagata 53, IS-107 Reykjavik, Iceland Chulalongkorn Univ, Fac Pharmaceut Sci, Dept Imaging Technol, 254 Payathai Rd, Bangkok 10330, ThailandStefansson, Einar论文数: 0 引用数: 0 h-index: 0机构: Landspitali Univ Hosp, Dept Ophthalmol, IS-101 Reykjavik, Iceland Chulalongkorn Univ, Fac Pharmaceut Sci, Dept Imaging Technol, 254 Payathai Rd, Bangkok 10330, Thailand
- [7] Macrocyclization: Enhancing Drug-like Properties of Discoidin Domain Receptor Kinase InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2025,Carzaniga, Laura论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, Italy Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, ItalyMazzucato, Roberta论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, Italy Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, ItalyMileo, Valentina论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, Italy Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, ItalyRizzi, Andrea论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, Italy Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, ItalyVallaro, Maura论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Mol Biotechnol & Hlth Sci Dept, CASS MedChem, I-10126 Turin, Italy Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, ItalyErmondi, Giuseppe论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Mol Biotechnol & Hlth Sci Dept, CASS MedChem, I-10126 Turin, Italy Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, ItalyCattani, Silvia论文数: 0 引用数: 0 h-index: 0机构: Univ Parma, Dept Chem Life Sci & Environm Sustainabil, I-43123 Parma, Italy Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, ItalySecchi, Andrea论文数: 0 引用数: 0 h-index: 0机构: Univ Parma, Dept Chem Life Sci & Environm Sustainabil, I-43123 Parma, Italy Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, ItalyCaron, Giulia论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Mol Biotechnol & Hlth Sci Dept, CASS MedChem, I-10126 Turin, Italy Chiesi Farmaceut, Corp Preclin R&D, Res Ctr, I-43122 Parma, Italy
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