Synthesis of thiazole-containing amino acids based on asparagine

被引：3
|
作者：
Bunev, A. S. [1 ]
Rudakova, Ya. I. [1 ]
Peregudov, A. S. [2 ]
Ostapenko, G. I. [1 ]
机构：
[1] Togliatti State Univ, Tolyatti 445667, Russia
[2] Russian Acad Sci, AN Nesmeyanov Organoelement Cpds Inst, Moscow 119991, Russia
来源：
RUSSIAN CHEMICAL BULLETIN | 2014年 / 63卷 / 05期
关键词：
amino acids; thiazoles; thioamides; Hantzsch synthesis; protecting groups; BIOLOGICAL EVALUATION; LARGAZOLE; INHIBITORS; OXAZOLE; DESIGN; POTENT;
D O I：
10.1007/s11172-014-0579-6
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A number of earlier unknown thiazole-containing amino acids were obtained by the Hantzsch reaction through the sequential transformation of asparagine to thio analog with subsequent reaction with alpha-bromoketones.
引用
收藏
页码：1232 / 1234
页数：3
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