One-pot synthesis of β-imidazolylpropionamides

被引：0
|
作者：
Ryabukhin, Sergey V. [1 ,2 ]
Granat, Dmitry S. [1 ]
Khodakovskiy, Pavel V. [1 ,2 ]
Shivanyuk, Alexander N. [1 ,2 ]
Tolmachev, Andrey A. [2 ]
机构：
[1] Enamine Ltd, UA-01103 Kiev, Ukraine
[2] Natl Taras Shevchenko Univ, UA-01033 Kiev, Ukraine
来源：
TETRAHEDRON LETTERS | 2008年 / 49卷 / 25期
关键词：
beta-imidazolylpropionamides; carbonyldiimidazole (CDI); acylation; acrylic acids;
D O I：
10.1016/j.tetlet.2008.04.096
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
New efficient one-pot methodology for the preparative synthesis of beta-imidazolylpropionamides was elaborated. It is based on the addition of imidazole to the activated double bond of the intermediate acrylimidazolide in the reaction between diverse acrylic acids and different amines promoted by CDI. A set of structurally and functionally diverse beta-imidazolylpropionamides was obtained in high preparative yields. (C) 2008 Elsevier Ltd. All rights reserved.
引用
收藏
页码：3997 / 4002
页数：6
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