Synthesis of advanced intermediates for the preparation of aza-analogues of podophyllotoxin

被引：23
|
作者：
Marcantoni, E [1 ]
Petrini, M [1 ]
Profeta, R [1 ]
机构：
[1] Univ Camerino, Dipartimento Sci Chim, I-62032 Camerino, Italy
来源：
TETRAHEDRON LETTERS | 2004年 / 45卷 / 10期
关键词：
Garner aldehyde; iminium ions; oxazolidinones; podophyllototin; sulfones;
D O I：
10.1016/j.tetlet.2004.01.040
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Some central intermediates useful for the synthesis of aza-analogues of the anti-carrier drug podophyllotoxin have been prepared starting from L-DOPA and (R)-Garner aldehyde. (C) 2001 Elsevier Ltd. All rights reserved.
引用
收藏
页码：2133 / 2136
页数：4
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