Prediction of blood-brain barrier penetration

被引:0
|
作者
Jorgensen, FS [1 ]
Jensen, LH [1 ]
Capion, D [1 ]
Christensen, IT [1 ]
机构
[1] Royal Danish Sch Pharm, Dept Med Chem, DK-2100 Copenhagen, Denmark
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:281 / 285
页数:5
相关论文
共 50 条
  • [1] Blood-brain barrier penetration prediction enhanced by uncertainty estimation
    Tong, Xiaochu
    Wang, Dingyan
    Ding, Xiaoyu
    Tan, Xiaoqin
    Ren, Qun
    Chen, Geng
    Rong, Yu
    Xu, Tingyang
    Huang, Junzhou
    Jiang, Hualiang
    Zheng, Mingyue
    Li, Xutong
    [J]. JOURNAL OF CHEMINFORMATICS, 2022, 14 (01)
  • [2] THE PREDICTION OF BLOOD-BRAIN BARRIER PENETRATION FOR MOLECULAR IMAGING AGENTS
    Newington, Ian M.
    Nairne, R. James D.
    Wynn, Duncan G.
    [J]. DRUGS OF THE FUTURE, 2009, 34 : 86 - 86
  • [3] Prediction of blood-brain barrier penetration: are we missing the point?
    Martin, I
    [J]. DRUG DISCOVERY TODAY, 2004, 9 (04) : 161 - 162
  • [4] Prediction of intestinal absorption and blood-brain barrier penetration by computational methods
    Clark, DE
    [J]. COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING, 2001, 4 (06) : 477 - 496
  • [5] Strategies to assess blood-brain barrier penetration
    Di, Li
    Kerns, Edward H.
    Carter, Guy T.
    [J]. EXPERT OPINION ON DRUG DISCOVERY, 2008, 3 (06) : 677 - 687
  • [6] PENETRATION OF BLOOD-BRAIN BARRIER BY METRONIDAZOLE AND TINIDAZOLE
    JOKIPII, AMM
    MYLLYLA, VV
    HOKKANEN, E
    JOKIPII, L
    [J]. JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY, 1977, 3 (03) : 239 - 245
  • [7] PENETRATION OF CATECHOLAMINES THROUGH BLOOD-BRAIN BARRIER
    ZAKUSOV, VV
    TOLMACHE.NS
    VYSOTSKA.NB
    [J]. BIULLETEN EKSPERIMENTALNOL BIOLOGII I MEDITSINY, 1972, 73 (05): : 64 - &
  • [8] Penetration of Intact Blood-Brain Barrier by Doripenem
    Margetis, K.
    Dimaraki, E.
    Charkoftaki, G.
    Vryonis, E.
    Markantonis, S.
    Boutos, N.
    Archontaki, H.
    Sakas, D. E.
    Valsami, G.
    Skoutelis, A.
    [J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2011, 55 (07) : 3637 - 3638
  • [9] PENETRATION OF SUGARS ACROSS BLOOD-BRAIN BARRIER
    EIDELBERG, E
    FISHMAN, J
    HAMS, ML
    [J]. JOURNAL OF PHYSIOLOGY-LONDON, 1967, 191 (01): : 47 - +
  • [10] PENETRATION OF CATECHOLAMINES THROUGH BLOOD-BRAIN BARRIER
    ZAKUSOV, VV
    VYSOTSKAYA, NB
    TOLMACHEVA, NS
    [J]. BULLETIN OF EXPERIMENTAL BIOLOGY AND MEDICINE,USSR, 1972, 73 (05): : 547 - +