共 50 条
- [1] Discovery of a Series of Pyrimidine Carboxamides as Inhibitors of Vanin-1[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (01) : 757 - 784Casimiro-Garcia, Agustin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAAllais, Christophe论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USABrennan, Agnes论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Inflammat & Immunol Res Unit, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAChoi, Chulho论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USADower, Gabriela论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Inflammat & Immunol Res Unit, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAFarley, Kathleen A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USAFleming, Margaret论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Inflammat & Immunol Res Unit, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAFlick, Andrew论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USAFrisbie, Richard K.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USAHall, Justin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USAHepworth, David论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAJones, Hannah论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAKnafels, John D.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USAKortum, Steve论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USALovering, Frank E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAMathias, John P.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAMohan, Sashi论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Inflammat & Immunol Res Unit, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAMorgan, Paul M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Inflammat & Immunol Res Unit, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAParng, Chuenlei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAParris, Kevin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USAPullen, Nick论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Inflammat & Immunol Res Unit, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USASchlerman, Franklin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Inflammat & Immunol Res Unit, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAStansfield, John论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Early Clin Dev Nonclin Stat, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAStrohbach, Joseph W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAVajdos, Felix F.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USAVincent, Fabien论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USAWang, Hong论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USAWang, Xiaolun论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAWebster, Robert论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Cambridge, MA 02139 USA Pfizer Inc, Med Design, Groton, CT 06340 USAWright, Stephen W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Med Design, Groton, CT 06340 USA Pfizer Inc, Med Design, Groton, CT 06340 USA
- [2] Visualization-Based Discovery of Vanin-1 Inhibitors for Colitis[J]. FRONTIERS IN CHEMISTRY, 2022, 9Wang, Guankai论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Cheeloo Coll Med,Key Lab Chem Biol MOE, Jinan, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Cheeloo Coll Med,Key Lab Chem Biol MOE, Jinan, Peoples R ChinaWang, Jingjing论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Cheeloo Coll Med,Key Lab Chem Biol MOE, Jinan, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Cheeloo Coll Med,Key Lab Chem Biol MOE, Jinan, Peoples R ChinaDu, Lupei论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Cheeloo Coll Med,Key Lab Chem Biol MOE, Jinan, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Cheeloo Coll Med,Key Lab Chem Biol MOE, Jinan, Peoples R ChinaLi, Minyong论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Cheeloo Coll Med,Key Lab Chem Biol MOE, Jinan, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Cheeloo Coll Med,Key Lab Chem Biol MOE, Jinan, Peoples R China
- [3] Discovery of a novel series of pyridine and pyrimidine carboxamides as potent and selective covalent inhibitors of Btk[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 28 (21) : 3419 - 3424Caldwell, Richard论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USALiu-Bujalski, Lesley论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAQiu, Hui论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAMochalkin, Igor论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAJones, Reinaldo论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USANeagu, Constantin论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAGoutopoulos, Andreas论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAGrenningloh, Roland论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAJohnson, Theresa论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USASherer, Brian论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAGardberg, Anna论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAFollis, Ariele Viacava论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAMorandi, Federica论文数: 0 引用数: 0 h-index: 0机构: L Hoffmann La Roche AG, Konzern Hauptsitz, Grenzacherstr 124, CH-4070 Basel, Switzerland EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USAHead, Jared论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45A Middlesex Turnpike, Billerica, MA 01821 USA
- [4] Discovery and characterization of dual inhibitors of human Vanin-1 and Vanin-2 enzymes through molecular docking and dynamic simulation-based approach[J]. INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2022, 213 : 1088 - 1097Nawaz, Muhammad Zohaib论文数: 0 引用数: 0 h-index: 0机构: Jiangsu Univ, Biofuels Inst, Sch Environm & Safety Engn, Zhenjiang 212013, Jiangsu, Peoples R ChinaAttique, Syed Awais论文数: 0 引用数: 0 h-index: 0机构: Univ Agr Faisalabad, Dept Comp Sci, Faisalabad 38040, Pakistan Jiangsu Univ, Biofuels Inst, Sch Environm & Safety Engn, Zhenjiang 212013, Jiangsu, Peoples R ChinaAin, Qurat-ul论文数: 0 引用数: 0 h-index: 0机构: Univ Sci & Technol China, Sch Life Sci, Hefei 230027, Peoples R China Jiangsu Univ, Biofuels Inst, Sch Environm & Safety Engn, Zhenjiang 212013, Jiangsu, Peoples R ChinaAlghamdi, Huda Ahmed论文数: 0 引用数: 0 h-index: 0机构: King Khalid Univ, Coll Sci, Dept Biol, Abha 61413, Saudi Arabia Jiangsu Univ, Biofuels Inst, Sch Environm & Safety Engn, Zhenjiang 212013, Jiangsu, Peoples R ChinaBilal, Muhammad论文数: 0 引用数: 0 h-index: 0机构: Huaiyin Inst Technol, Sch Life Sci & Food Engn, Huaian, Peoples R China Jiangsu Univ, Biofuels Inst, Sch Environm & Safety Engn, Zhenjiang 212013, Jiangsu, Peoples R ChinaYan, Wei论文数: 0 引用数: 0 h-index: 0机构: China Univ Geosci, Coll Marine Sci & Technol, Dept Marine Sci, Wuhan, Peoples R China Jiangsu Univ, Biofuels Inst, Sch Environm & Safety Engn, Zhenjiang 212013, Jiangsu, Peoples R China论文数: 引用数: h-index:机构:
- [5] Influence of Vanin-1 and Catalytic Products in Liver During Normal and Oxidative Stress Conditions[J]. CURRENT MEDICINAL CHEMISTRY, 2015, 22 (20) : 2407 - 2416Ferreira, Daniel W.论文数: 0 引用数: 0 h-index: 0机构: Univ Connecticut, Dept Pharmaceut Sci, Storrs, CT 06269 USA Univ Connecticut, Dept Pharmaceut Sci, Storrs, CT 06269 USANaquet, Philippe论文数: 0 引用数: 0 h-index: 0机构: Aix Marseille Univ, CNRS, INSERM, CIML, Marseille, France Univ Connecticut, Dept Pharmaceut Sci, Storrs, CT 06269 USAManautou, Jose E.论文数: 0 引用数: 0 h-index: 0机构: Univ Connecticut, Dept Pharmaceut Sci, Storrs, CT 06269 USA Univ Connecticut, Dept Pharmaceut Sci, Storrs, CT 06269 USA
- [6] Design, synthesis, and evaluation of new vanin-1 inhibitors based on RR6[J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 65Yoneyama, Hiroki论文数: 0 引用数: 0 h-index: 0机构: Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, Japan Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, JapanHosohata, Keiko论文数: 0 引用数: 0 h-index: 0机构: Osaka Med & Pharmaceut Univ, Fac Pharm, Educ & Res Ctr Clin Pharm, 4-20-1Nasahara, Takatsuki, Osaka 5691094, Japan Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, JapanJin, Denan论文数: 0 引用数: 0 h-index: 0机构: Osaka Med & Pharmaceut Univ, Grad Sch Med, Dept Innovat Med, 2-7 Daigaku Machi, Takatsuki, Osaka 5698686, Japan Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, JapanYoshida, Iroha论文数: 0 引用数: 0 h-index: 0机构: Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, Japan Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, JapanToyoda, Miyui论文数: 0 引用数: 0 h-index: 0机构: Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, Japan Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, JapanKitamura, Ikuko论文数: 0 引用数: 0 h-index: 0机构: Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, Japan Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, JapanTakai, Shinji论文数: 0 引用数: 0 h-index: 0机构: Osaka Med & Pharmaceut Univ, Grad Sch Med, Dept Innovat Med, 2-7 Daigaku Machi, Takatsuki, Osaka 5698686, Japan Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, JapanUsami, Yoshihide论文数: 0 引用数: 0 h-index: 0机构: Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, Japan Osaka Med & Pharmaceut Univ, Fac Pharm, Dept Pharmaceut Organ Chem, 4-20-1Nasahara, Takatsuki, Osaka 5691094, Japan
- [7] Vanin-1 expression and methylation discriminate pediatric asthma corticosteroid treatment response[J]. JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY, 2015, 136 (04) : 923 - +Xiao, Chang论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAMyers, Jocelyn M. Biagini论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAJi, Hong论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAMetz, Kelly论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Allergy & Immunol, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAMartin, Lisa J.论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Human Genet, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USALindsey, Mark论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAHe, Hua论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Human Genet, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAPowers, Racheal论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAUlm, Ashley论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USARuff, Brandy论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAEricksen, Mark B.论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USASomineni, Hari K.论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USASimmons, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Hosp Med, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAStrait, Richard T.论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Emergency Med, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAKercsmar, Carolyn M.论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Pulm Med, Cincinnati, OH USA Univ Cincinnati, Dept Pediat, Cincinnati Childrens Hosp Med Ctr, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USAHershey, Gurjit K. Khurana论文数: 0 引用数: 0 h-index: 0机构: Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA Univ Cincinnati, Cincinnati Childrens Hosp Med Ctr, Div Asthma Res, Cincinnati, OH USA
- [8] Early Process Development of Two Vanin-1 Inhibitors: Solid Form Challenges and Control of Ambident Reactivity[J]. ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2024, 28 (06) : 2226 - 2236Allais, Christophe论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USACasimiro-Garcia, Agustin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Cambridge, MA 02142 USA Pfizer Res & Dev, Groton, CT 06340 USADion, Amelie论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USAJensen, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USAKeene, Nandell论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USAKumar, Rajesh论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USALi, Bryan论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USALall, Manjinder S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USAMcwilliams, J. Christopher论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USAWood, Geoffrey P. F.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USAWright, Stephen W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USAYu, Shu论文数: 0 引用数: 0 h-index: 0机构: Pfizer Res & Dev, Groton, CT 06340 USA Pfizer Res & Dev, Groton, CT 06340 USA
- [9] Discovery of pyrimidine carboxamides as potent and selective CCK1 receptor agonists[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (10) : 2911 - 2915Wang, Liping论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAHubert, James A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Pharmacol, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USALee, Susan J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Pharmacol, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAPan, Jie论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Metab Disorders, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAQian, Su论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Metab Disorders, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAReitman, Marc L.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Metab Disorders, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAStrack, Alison M.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Pharmacol, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAWeingarth, Drew T.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Metab Disorders, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAMacNeil, Douglas J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Metab Disorders, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAWeber, Ann E.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAEdmondson, Scott D.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USA
- [10] Discovery of diaminotriazine carboxamides as potent inhibitors of hematopoetic progenitor kinase 1[J]. BIOORGANIC CHEMISTRY, 2023, 138Zhou, Lixin论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R ChinaYe, Xiuquan论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R ChinaWang, Kaizhen论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R ChinaShen, Hongtao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R ChinaWang, Tianyu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R ChinaZhang, Xiangyu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R ChinaJiang, Sheng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R ChinaXiao, Yibei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R ChinaZhang, Kuojun论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 210009, Peoples R China