Synthesis and antifungal activity of novel 3,6-Diaryl-5H[1,2,4]triazolo[4,3-b][1,2,4]triazepines

被引:12
|
作者
Gupta, Monika [1 ]
机构
[1] Univ Jammu, Dept Chem, Jammu 180006, India
关键词
D O I
10.1002/jhet.5570440508
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
5-Aryl-3,4-diamino-1,2,4-triazoles 5 on treatment with beta-chlorocinnamaldehydes 7 in the presence of catalytic amount of p-TsOH and N,N-dimethylformamide as an energy transfer medium under microwave irradiation and as solvent with oil-bath heating at 80 degrees C affords novel 3,6-diaryl-5H-[1,2,4]triazolo[4,3-b]-1,2,4]triazepines 8. The structures of the synthesized compounds were established on the basis of H-1 NMR, IR, mass spectral data and elemental analysis.
引用
收藏
页码:1023 / 1027
页数:5
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