Discovery and development of covalent BTK inhibitors

被引:0
|
作者
Chen, Wei [1 ]
机构
[1] Pharmacyclics Inc, Sunnyvale, CA USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
204
引用
收藏
页数:1
相关论文
共 50 条
  • [1] The Role of Noncovalent BTK Inhibitors in the Era of Covalent BTK Inhibitors
    Qan, Fateeha Fur
    Shah, Nirav N.
    [J]. CLINICAL ADVANCES IN HEMATOLOGY & ONCOLOGY, 2024, 22 (03) : 140 - 147
  • [2] Discovery and development of CC-292, a covalent inhibitor of BTK
    Petter, Russell
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250
  • [3] Considerations in the generation of covalent BTK inhibitors
    Wilson, Noel
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 256
  • [4] Covalent Inhibitors of BTK in the Treatment of CLL
    Woyach, Jennifer A.
    [J]. CLINICAL LYMPHOMA MYELOMA & LEUKEMIA, 2023, 23 : S31 - S32
  • [5] Discovery of a Novel Class of Covalent Dual Inhibitors Targeting the Protein Kinases BMX and BTK
    Forster, Michael
    Liang, Xiaojun Julia
    Schroeder, Martin
    Gerstenecker, Stefan
    Chaikuad, Apirat
    Knapp, Stefan
    Laufer, Stefan
    Gehringer, Matthias
    [J]. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2020, 21 (23) : 1 - 36
  • [6] Discovery of a novel series of pyridine and pyrimidine carboxamides as potent and selective covalent inhibitors of Btk
    Caldwell, Richard
    Liu-Bujalski, Lesley
    Qiu, Hui
    Mochalkin, Igor
    Jones, Reinaldo
    Neagu, Constantin
    Goutopoulos, Andreas
    Grenningloh, Roland
    Johnson, Theresa
    Sherer, Brian
    Gardberg, Anna
    Follis, Ariele Viacava
    Morandi, Federica
    Head, Jared
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 28 (21) : 3419 - 3424
  • [7] Discovery of potent, highly selective covalent irreversible BTK inhibitors from a fragment hit
    Qiu, Hui
    Liu-Bujalski, Lesley
    Caldwell, Richard D.
    Follis, Ariele Viacava
    Gardberg, Anna
    Goutopoulos, Andreas
    Grenningloh, Roland
    Head, Jared
    Johnson, Theresa
    Jones, Reinaldo
    Mochalkin, Igor
    Morandi, Federica
    Neagh, Constantin
    Sherer, Brian
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 28 (17) : 2939 - 2944
  • [8] An update on the discovery and development of reversible covalent inhibitors
    Faridoon
    Ng, Raymond
    Zhang, Guiping
    Li, Jie Jack
    [J]. MEDICINAL CHEMISTRY RESEARCH, 2023, 32 (06) : 1039 - 1062
  • [9] An update on the discovery and development of reversible covalent inhibitors
    Raymond Faridoon
    Guiping Ng
    Jie Jack Zhang
    [J]. Medicinal Chemistry Research, 2023, 32 : 1039 - 1062
  • [10] Drug discovery considerations in the development of covalent inhibitors
    Mah, Robert
    Thomas, Jason R.
    Shafer, Cynthia M.
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (01) : 33 - 39