Minimization of potential hERG liability in histamine H3 receptor antagonists

被引：14
|
作者：
Black, L. A. [1 ]
Liu, H. [1 ]
Diaz, G. J. [1 ]
Fox, G. B. [1 ]
Browman, K. E. [1 ]
Wetter, J. [1 ]
Marsh, K. C. [1 ]
Miller, T. R. [1 ]
Esbenshade, T. A. [1 ]
Brioni, J. [1 ]
Cowart, M. D. [1 ]
机构：
[1] Abbott Labs, GPRD Neurosci Res, Abbott Pk, IL 60064 USA
来源：
INFLAMMATION RESEARCH | 2008年 / 57卷 / Suppl 1期
关键词：
Benzofuran; Dofetilide; hERG Channel; Selectivity Ratio; Cyanophenyl;
D O I：
10.1007/s00011-007-0622-2
中图分类号：
Q2 [细胞生物学];
学科分类号：
071009 ; 090102 ;
摘要：
引用
收藏
页码：S45 / S46
页数：2
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