Facile synthesis of methyl 2-amino-3-(2-methyl-3-quinolyl)propanoate

被引：6
|
作者：
Hadden, M [1 ]
Stevenson, PJ [1 ]
机构：
[1] Queens Univ Belfast, Sch Chem, Belfast BT9 5AG, Antrim, North Ireland
来源：
JOURNAL OF CHEMICAL RESEARCH | 1998年 / 12期
关键词：
D O I：
10.1039/a804962i
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Methyl 4-acetyl-5-(2-nitrophenyl)pyrrolidine-2-carboxylate 5, readily available in one step by a 1,3-dipolar cycloaddition, undergoes reduction, cyclisation and fragmentation to the corresponding quinoline when treated with hydrogen and palladium.
引用
收藏
页码：796 / 797
页数：3
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