(2,3-Dihydro-1H-indol-5-ylmethyl)amine

被引：0
|
作者：
Ogurtsov, Vladimir A. [1 ]
Rakitin, Oleg A. [1 ,2 ]
机构：
[1] Russian Acad Sci, ND Zelinsky Inst Organ Chem, 47 Leninsky Prospekt, Moscow 119991, Russia
[2] South Ural State Univ, Nanotechnol Educ & Res Ctr, 76 Lenina Ave, Chelyabinsk 454080, Russia
来源：
MOLBANK | 2021年 / 2021卷 / 03期
关键词：
2,3-dihydroindoles (indolines); (2,3-dihydro-1H-indol-5-ylmethyl)amine; deprotection; biological activity;
D O I：
10.3390/M1248
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
New (2,3-dihydro-1H-indol-5-ylmethyl)amine was synthesized from 2-((1-acetylindolin-5-yl)methyl)isoindoline-1,3-dione by simultaneous deprotection of phthalimide and acetyl groups. The structure of the newly synthesized compounds was established by elemental analysis, high resolution mass-spectrometry, H-1, C-13 NMR and IR spectroscopy and mass-spectrometry. The resulting compound is a convenient intermediate for various disubstituted 1-(indolin-5-yl)methanamines, which may be of interest as substances with useful pharmacological properties.
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页数：3
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