MEDI 269-Computational neural network analysis of the affinity of lobeline and tetrabenazine analogs for the vesicular monoamine transporter-2

被引：0

作者：

Cox, Christopher D. ^{[1
]}

Coleman, Paul J. ^{[1
]}

Fraley, Mark E. ^{[1
]}

Garbaccio, Robert M. ^{[1
]}

Breslin, Michael J. ^{[1
]}

Whitman, David B. ^{[1
]}

Schreier, John D. ^{[1
]}

Hartman, George D. ^{[1
]}

Torrent, Maricel ^{[2
]}

Lobell, Rob ^{[3
]}

Buser, Carolyn ^{[3
]}

Tao, Weikang ^{[3
]}

Huber, Hans ^{[3
]}

Kohl, Nancy E. ^{[3
]}

Yan, Youwei ^{[4
]}

Kuo, Lawrence C. ^{[4
]}

机构：

[1] Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

[2] Merck & Co Inc, Dept Mol Syst, West Point, PA 19486 USA

[3] Merck & Co Inc, Dept Canc Res, West Point, PA 19486 USA

[4] Merck & Co Inc, Dept Biol Struct, West Point, PA 19486 USA

来源：

ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2007年 / 233卷

关键词：

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

211-MEDI

引用

页码：960 / 960

页数：1

共 13 条

[1] Computational neural network analysis of the affinity of lobeline and tetrabenazine analogs for the vesicular monoamine transporter-2
Zheng, Fang
Zheng, Guangrong
Deaciuc, A. Gabriela
Zhan, Chang-Guo
Dwoskin, Linda P.
Crooks, Peter A.
BIOORGANIC & MEDICINAL CHEMISTRY, 2007, 15 (08) : 2975 - 2992
[2] Computational neural network analysis of the affinity of lobeline and tetrabenazine analogs for the vesicular monoamine transporter-2
Zheng, Fang
Zheng, Guangrong
Deaciuc, A. Gabriela
Zhan, Chang-Guo
Dwoskin, Linda P.
Crooks, Peter A.
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 233 : 844 - 844
[3] Design, Synthesis and Interaction at the Vesicular Monoamine Transporter-2 of Lobeline Analogs: Potential Pharmacotherapies for the Treatment of Psychostimulant Abuse
Crooks, Peter A.
Zheng, Guangrong
Vartak, Ashish P.
Culver, John P.
Zheng, Fang
Horton, David B.
Dwoskin, Linda P.
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2011, 11 (09) : 1103 - 1127
[4] Kinetic analysis of developmental changes in vesicular monoamine transporter-2 function
Volz, Trent J.
Hanson, Glen R.
Fleckenstein, Annette E.
SYNAPSE, 2006, 60 (06) : 474 - 477
[5] Pyrrolidine analogs of GZ-793A: Synthesis and evaluation as inhibitors of the vesicular monoamine transporter-2 (VMAT2)
Penthala, Narsimha Reddy
Ponugoti, Purushothama Rao
Nickell, Justin R.
Deaciuc, Agripina G.
Dwoskin, Linda P.
Crooks, Peter A.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (11) : 3342 - 3345
[6] meso-Transdiene Analogs Inhibit Vesicular Monoamine Transporter-2 Function and Methamphetamine-Evoked Dopamine Release
Horton, David B.
Siripurapu, Kiran B.
Norrholm, Seth D.
Culver, John P.
Hojahmat, Marhaba
Beckmann, Joshua S.
Harrod, Steven B.
Deaciuc, Agripina G.
Bardo, Michael T.
Crooks, Peter A.
Dwoskin, Linda P.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2011, 336 (03): : 940 - 951
[7] Phenyl Ring-Substituted Lobelane Analogs: Inhibition of [3H]Dopamine Uptake at the Vesicular Monoamine Transporter-2
Nickell, Justin R.
Zheng, Guangrong
Deaciuc, Agripina G.
Crooks, Peter A.
Dwoskin, Linda P.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2011, 336 (03): : 724 - 733
[8] Synthesis and in vitro evaluation of water-soluble 1,4-diphenethylpiperazine analogs as novel inhibitors of the vesicular monoamine transporter-2
Nickell, Justin R.
Culver, John P.
Janganati, Venumadhav
Zheng, Guangrong
Dwoskin, Linda P.
Crooks, Peter A.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 26 (18) : 4441 - 4445
[9] Tetrabenazine, a vesicular monoamine transporter-2 inhibitor, attenuates morphine-induced hyperlocomotion in mice through alteration of dopamine and 5-hydroxytryptamine turnover in the cerebral cortex
Kitanaka, Nobue
Kitanaka, Junichi
Hall, F. Scott
Kandori, Takashi
Murakami, Ayaka
Muratani, Kazuki
Nakano, Tae
Uhl, George R.
Takemura, Motohiko
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 2018, 172 : 9 - 16
[10] Novel N-1,2-Dihydroxypropyl Analogs of Lobelane Inhibit Vesicular Monoamine Transporter-2 Function and Methamphetamine-Evoked Dopamine Release
Horton, David B.
Siripurapu, Kiran B.
Zheng, Guangrong
Crooks, Peter A.
Dwoskin, Linda P.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2011, 339 (01): : 286 - 297

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