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- [1] Discovery of cell-active phenyl-imidazole Pin1 inhibitors by structure-guided fragment evolutionBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (22) : 6483 - 6488Potter, Andrew论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandOldfield, Victoria论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandNunns, Claire论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandFromont, Christophe论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandRay, Stuart论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandNorthfield, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandBryant, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandScrace, Simon F.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandRobinson, David论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandMatossova, Natalia论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandBaker, Lisa论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandDokurno, Pawel论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandSurgenor, Allan E.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandDavis, Ben论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandRichardson, Christine M.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandMurray, James B.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, EnglandMoore, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Vernalis R&D Ltd, Cambridge CB21 6GB, England
- [2] Fragment-based and structure-guided discovery of perforin inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 261论文数: 引用数: h-index:机构:Law, Ruby H. P.论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Dept Biochem & Mol Biol, Clayton, Vic 3800, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandLeung, Eleanor W. W.论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New Zealand论文数: 引用数: h-index:机构:Akhlaghi, Hedieh论文数: 0 引用数: 0 h-index: 0机构: Peter MacCallum Canc Ctr, Canc Immunol Program, 305 Grattan St, Melbourne, Vic 3000, Australia Univ Melbourne, Sir Peter MacCallum Dept Oncol, Parkville, Vic 3052, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandChandrashekaran, Indu R.论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia Monash Univ, ARC Ctr Fragment Based Design, Parkville, Vic 3052, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandCaradoc-Davies, Tom T.论文数: 0 引用数: 0 h-index: 0机构: Australian Synchrotron, 800 Blackburn Rd, Melbourne, Vic 3168, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New Zealand论文数: 引用数: h-index:机构:Feutrill, John论文数: 0 引用数: 0 h-index: 0机构: Synth Med Chem Australia Pty Ltd, Bio21 Inst, 30 Flemington Rd, Parkville, Vic 3052, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandMiddlemiss, David论文数: 0 引用数: 0 h-index: 0机构: XaviaPharm, Bishops Stortford CM23 3NF, England Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandJeevarajah, Devadharshini论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Dept Biochem & Mol Biol, Clayton, Vic 3800, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandBashtannyk-Puhalovich, Tanya论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Dept Biochem & Mol Biol, Clayton, Vic 3800, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandGiddens, Anna C.论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New Zealand Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandLee, Tet Woo论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New Zealand Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandJamieson, Stephen M. F.论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New Zealand New Zealand Ctr Res Excellence, Maurice Wilkins Ctr Mol Biodiscovery, Auckland, New Zealand Univ Auckland, Fac Med & Hlth Sci, Dept Pharmacol & Clin Pharmacol, Private Bag 92019, Auckland 1142, New Zealand Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandTrapani, Joseph A.论文数: 0 引用数: 0 h-index: 0机构: Peter MacCallum Canc Ctr, Canc Immunol Program, 305 Grattan St, Melbourne, Vic 3000, Australia Univ Melbourne, Sir Peter MacCallum Dept Oncol, Parkville, Vic 3052, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandWhisstock, James C.论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Dept Biochem & Mol Biol, Clayton, Vic 3800, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandSpicer, Julie A.论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New Zealand New Zealand Ctr Res Excellence, Maurice Wilkins Ctr Mol Biodiscovery, Auckland, New Zealand Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New ZealandNorton, Raymond S.论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia Monash Univ, ARC Ctr Fragment Based Design, Parkville, Vic 3052, Australia Univ Auckland, Fac Med & Hlth Sci, Auckland Canc Soc Res Ctr, Private Bag 92019, Auckland 1142, New Zealand
- [3] Fragment-Based and Structure-Guided Discovery and Optimization of Rho Kinase InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (05) : 2474 - 2478Li, Rongshi论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USAMartin, Mathew P.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USALiu, Yan论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USAWang, Binglin论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USAPatel, Ronil A.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USAZhu, Jin-Yi论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USASun, Nan论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USAPireddu, Roberta论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USALawrence, Nicholas J.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USALi, Jiannong论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Expt Therapeut, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USAHaura, Eric B.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Expt Therapeut, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USASung, Shen-Shu论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USAGuida, Wayne C.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USASchonbrunn, Ernst论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USASebti, Said M.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Drug Discovery, Tampa, FL 33612 USA
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- [5] Novel targets in oncology: Discovery of novel allosteric inhibitors of IRE1αABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 247Evans, Karen A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Dept Oncol R&D, Collegeville, PA 19426 USA GlaxoSmithKline, Dept Oncol R&D, Collegeville, PA 19426 USA
- [6] Aminoindazole PDK1 Inhibitors: A Case Study in Fragment-Based Drug DiscoveryACS MEDICINAL CHEMISTRY LETTERS, 2010, 1 (08): : 439 - 442Medina, Jesus R.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USABlackledge, Charles W.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USAHeerding, Pirk A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USACampobasso, Nino论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Mol Discovery Res, Computat & Struct Chem, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USAWard, Paris论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Mol Discovery Res, Computat & Struct Chem, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USABriand, Jacques论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Mol Discovery Res, Analyt Chem, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USAWright, Lois论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Mol Discovery Res, Screening & Compound Profiling, Res Triangle Pk, NC 27709 USA GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USAAxten, Jeffrey M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Oncol Res, Signal Transduct DPU Med Chem, Collegeville, PA 19426 USA
- [7] Structure-guided discovery of novel aminoglycoside mimetics as antibacterial translation inhibitorsANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2005, 49 (12) : 4942 - 4949Zhou, YF论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USAGregor, VE论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USASun, ZX论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USAAyida, BK论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USAWinters, GC论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USAMurphy, D论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USASimonsen, KB论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USAVourloumis, D论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USAFish, S论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USAFroelich, JM论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USAWall, D论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USAHermann, T论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USA
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