Design and Efficient Synthesis of Some Azole and Thiazole Systems Based 3-(1,3-Dioxoisoindolin-2-yl)-3-oxopropanenitrile

被引：0
|
作者：
El Aazab, Islam Helmy [1 ,2 ]
El Latif, Fawi Mohamed Abd [2 ]
机构：
[1] Aswan Univ, Fac Sci, Dept Chem, Aswan 81528, Egypt
[2] Taif Univ, Fac Sci, Dept Chem, At Taif 21974, Saudi Arabia
来源：
LETTERS IN ORGANIC CHEMISTRY | 2015年 / 12卷 / 03期
关键词：
Azole; thiazole; phthalimide; pyrazole; enaminonitrile; 1,3-dioxoisoindoline; ANTIMICROBIAL ACTIVITY; DERIVATIVES; CHEMISTRY; FACILE;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A variety of pyrazoles, thiazoles, thiadiazoles, thiazolidines, azetidine, thiazolo[3,2-a] pyrimidine and pyrazolo[3,4-b]pyridine systems, based on 3-(1,3-dioxoisoindolin-2-yl)-3-oxopropanenitrile precursor are synthesized in good yields. The mechanistic aspect for the formation of the newly synthesized compounds is discussed and the structure of the synthesized compounds was established based on elemental analysis and spectral data.
引用
收藏
页码：187 / 196
页数：10
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