An Efficient One-Pot Synthesis of 1, 5-Benzodiazepine Derivatives Catalyzed by TBAB under Mild Conditions

被引：4
|
作者：
Baseer, Mohammad A. [1 ]
Khan, Asgar Jafar [2 ]
机构：
[1] Yeshwant Mahavidyalaya, Organ Chem Res Lab, Nanded 431602, India
[2] Milliya Coll, Organ Synth Lab, Beed 431122, India
来源：
E-JOURNAL OF CHEMISTRY | 2012年 / 9卷 / 01期
关键词：
Tetra butyl ammonium bromide; 1; 5-Benzodiazepine; o-Phenylenediamine; Ketones; Short reaction time; 1,5-BENZODIAZEPINE DERIVATIVES; PROMOTED SYNTHESIS;
D O I：
10.1155/2012/657439
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
2,3-Dihydro-1H-1,5-benzodiazepines were synthesized by reaction of o-phenylenediamine with ketones (acyclic / cyclic) under solvent free conditions in the presence of tetra butyl ammonium bromide (TBAB) in short reaction time with excellent yield.
引用
收藏
页码：407 / 414
页数：8
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