Anti-atherosclerotic effect of the novel acyl-CoA:cholesterol acyltransferase inhibitor, K-10191, on high cholesterol-fed rabbits

被引:0
|
作者
Yoshinaka, Y [1 ]
Kobayashi, H [1 ]
Kawamine, K [1 ]
Shibuya, K [1 ]
Sato, F [1 ]
机构
[1] Kowa Co Ltd, Tokyo, Japan
关键词
D O I
10.1016/S1567-5688(03)90719-7
中图分类号
R6 [外科学];
学科分类号
1002 ; 100210 ;
摘要
引用
收藏
页码:166 / 167
页数:2
相关论文
共 50 条
  • [1] Plaque stabilization of the novel acyl-CoA:cholesterol acyltransferase inhibitor, K-10191, in apoE knockout mice
    Kobayashi, H
    Kawamine, K
    Yoshinaka, Y
    Shibuya, K
    Sato, F
    [J]. ATHEROSCLEROSIS SUPPLEMENTS, 2003, 4 (02) : 161 - 161
  • [2] Anti-atherosclerotic effect of E5324, an inhibitor of acyl-CoA:cholesterol acyltransferase, in Watanabe heritable hyperlipidemic rabbits
    Kogushi, M
    Tanaka, H
    Ohtsuka, I
    Yamada, T
    Kobayashi, H
    Saeki, T
    Takada, M
    Hiyoshi, H
    Yanagimachi, M
    Kimura, T
    Yoshitake, S
    Saito, I
    [J]. ATHEROSCLEROSIS, 1996, 124 (02) : 203 - 210
  • [3] NTE-122, an acyl-CoA:cholesterol acyltransferase inhibitor, prevents the progression of atherogenesis in cholesterol-fed rabbits
    Azuma, Y
    Date, K
    Ohno, K
    Matsushiro, S
    Nobuhara, Y
    Yamada, T
    [J]. JAPANESE JOURNAL OF PHARMACOLOGY, 2001, 86 (01): : 120 - 123
  • [4] Pharmacological properties of R-755, a novel acyl-CoA:cholesterol acyltransferase inhibitor, in cholesterol-fed rats, hamsters and rabbits
    Matsui, Y
    Horiuchi, K
    Yamamoto, K
    Kanai, K
    [J]. JAPANESE JOURNAL OF PHARMACOLOGY, 2001, 85 (04): : 423 - 433
  • [5] CONTROL OF HEPATIC ACYL-COA - CHOLESTEROL ACYLTRANSFERASE IN CHOLESTEROL-FED RATS
    HIGGINS, MJP
    PAPACHRISTODOULOU, DK
    [J]. BIOCHEMICAL SOCIETY TRANSACTIONS, 1989, 17 (01) : 156 - 156
  • [6] Anti-atherosclerotic effects of tamoxifen in cholesterol-fed ovariectomized rabbits
    Sugama, D
    Nakajima, H
    Maehara, K
    Hara, I
    Lawlor, GF
    Inazu, M
    Yamashina, A
    Matsumiya, T
    [J]. JAPANESE HEART JOURNAL, 2002, 43 (05): : 545 - 558
  • [7] Inhibitory effect of monatepil maleate on acyl-CoA:cholesterol acyltransferase activity in the liver of cholesterol-fed Japanese monkeys
    Sumiya, T
    Ikeno, A
    Kato, H
    Fujitani, B
    Masuda, Y
    Hosoki, K
    Miyazaki, M
    [J]. AMERICAN JOURNAL OF HYPERTENSION, 1997, 10 (07) : 779 - 785
  • [8] Effect of F-1394, an acyl-CoA:cholesterol acyltransferase inhibitor, on atherosclerosis induced by high cholesterol diet in rabbits
    Aragane, K
    Kojima, K
    Fujinami, K
    Kamei, J
    Kusunoki, J
    [J]. ATHEROSCLEROSIS, 2001, 158 (01) : 139 - 145
  • [9] Cholesterol-lowering effects of NTE-122, a novel acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor, on cholesterol diet-fed rats and rabbits
    Azuma, Y
    Kawasaki, T
    Ikemoto, K
    Obata, K
    Ohno, K
    Sajiki, N
    Yamada, T
    Yamasaki, M
    Nobuhara, Y
    [J]. JAPANESE JOURNAL OF PHARMACOLOGY, 1998, 78 (03): : 355 - 364
  • [10] Discovery of a Potent and Orally Available Acyl-CoA: Cholesterol Acyltransferase Inhibitor as an Anti-atherosclerotic Agent: (4-Phenylcoumarin)acetanilide Derivatives
    Ogino, Masaki
    Fukui, Seiji
    Nakada, Yoshihisa
    Tokunoh, Ryosuke
    Itokawa, Shigekazu
    Kakoi, Yuichi
    Nishimura, Satoshi
    Sanada, Tsukasa
    Fuse, Hiromitsu
    Kubo, Kazuki
    Wada, Takeo
    Marui, Shogo
    [J]. CHEMICAL & PHARMACEUTICAL BULLETIN, 2011, 59 (10) : 1268 - 1273