Design, green synthesis, anti-microbial, and anti-oxidant activities of novel α-aminophosphonates via Kabachnik-Fields reaction

被引：24

作者：

Sampath, C. ^{[1
]}

Harika, P. ^{[2
]}

Revaprasadu, N. ^{[1
]}

机构：

[1] Univ Zululand, Dept Chem, ZA-3886 Kwa Dlangezwa, Kwazulu Natal, South Africa

[2] Andhra Loyola Inst Engn & Technol, Dept Chem, Vijayawada, Andhra Pradesh, India

来源：

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 2016年 / 191卷 / 08期

基金：

新加坡国家研究基金会;

关键词：

alpha-Aminophosphonates; Kabachnik-Fields reaction; green synthesis; anti-microbial activity; anti-oxidant activity; BIOLOGICAL-ACTIVITY; AMINO PHOSPHONATES; ACID;

D O I：

10.1080/10426507.2015.1035379

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

An efficient and environmentally friendly protocol has been developed for the synthesis of novel -aminophosphonates in good to excellent yields (76-92%) by a one-pot, three-component reaction of an amine, an aldehyde, and diphenyl phosphite using polyethylene glycol (PEG-400) as a green solvent at 80 degrees C via Kabachnik-Fields reaction. Their chemical structures were elucidated by IR, H-1, C-13, and P-31 NMR spectroscopy, mass spectrometry, and elemental analysis. The titled compounds displayed moderate to high anti-microbial and anti-oxidant activities.

引用

页码：1081 / 1085

页数：5

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