Multitarget Drug Discovery and Polypharmacology

被引:157
|
作者
Bolognesi, Maria Laura [1 ]
Cavalli, Andrea [1 ,2 ]
机构
[1] Univ Bologna, Alma Mater Studiorum, Dipartimento Farm & Biotecnol, Via Belmeloro 6, I-40126 Bologna, Italy
[2] Ist Italiano Tecnol, CompuNet, Via Morego 30, I-16163 Genoa, Italy
关键词
ALZHEIMERS-DISEASE; INHIBITORS;
D O I
10.1002/cmdc.201600161
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:1190 / 1192
页数:3
相关论文
共 50 条
  • [1] Polypharmacology in a Single Drug: Multitarget Drugs
    Bolognesi, M. L.
    [J]. CURRENT MEDICINAL CHEMISTRY, 2013, 20 (13) : 1639 - 1645
  • [2] Polypharmacology in Drug Discovery
    Scotti, Luciana
    Scotti, Marcus T.
    [J]. CURRENT PHARMACEUTICAL DESIGN, 2016, 22 (21) : 3071 - 3072
  • [3] Polypharmacology: drug discovery for the future
    Reddy, A. Srinivas
    Zhang, Shuxing
    [J]. EXPERT REVIEW OF CLINICAL PHARMACOLOGY, 2013, 6 (01) : 41 - 47
  • [4] Systems approaches to polypharmacology and drug discovery
    Boran, Aislyn D. W.
    Iyengar, Ravi
    [J]. CURRENT OPINION IN DRUG DISCOVERY & DEVELOPMENT, 2010, 13 (03) : 297 - 309
  • [5] Polypharmacology: Challenges and Opportunities in Drug Discovery
    Anighoro, Andrew
    Bajorath, Juergen
    Rastelli, Giulio
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (19) : 7874 - 7887
  • [6] Computational polypharmacology: a new paradigm for drug discovery
    Chaudhari, Rajan
    Tan, Zhi
    Huang, Beibei
    Zhang, Shuxing
    [J]. EXPERT OPINION ON DRUG DISCOVERY, 2017, 12 (03) : 279 - 291
  • [7] AI for targeted polypharmacology: The next frontier in drug discovery
    Cichonska, Anna
    Ravikumar, Balaguru
    Rahman, Rayees
    [J]. CURRENT OPINION IN STRUCTURAL BIOLOGY, 2024, 84
  • [8] Polypharmacology in Drug Discovery: A Review from Systems Pharmacology Perspective
    Zhang, Wenjuan
    Bai, Yaofei
    Wang, Yonghua
    Xiao, Wei
    [J]. CURRENT PHARMACEUTICAL DESIGN, 2016, 22 (21) : 3171 - 3181
  • [9] Predicting Targeted Polypharmacology for Drug Repositioning and Multi-Target Drug Discovery
    Liu, X.
    Zhu, F.
    Ma, X. H.
    Shi, Z.
    Yang, S. Y.
    Wei, Y. Q.
    Chen, Y. Z.
    [J]. CURRENT MEDICINAL CHEMISTRY, 2013, 20 (13) : 1646 - 1661
  • [10] Polypharmacology, drug repurposing and collaborative drug discovery: Shining light or flash in the pan?
    Lipinski, Christopher A.
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 243