One step synthesis of 4-arylpolyhydroquinoline derivatives using microwave irradiation

被引:0
|
作者
Tu, SJ [1 ]
Zhou, JF [1 ]
Deng, X [1 ]
Cai, PJ [1 ]
Wang, H [1 ]
Feng, JC [1 ]
机构
[1] Nanjing Univ, Dept Chem, Nanjing 210093, Peoples R China
关键词
polyhydroquinoline derivative; synthesis; microwave irradiation;
D O I
暂无
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A series of 4-aryl-3-ethoxylcarbonyl-1, 4, 5, 6, 7, 8-hexahydro-5-oxo-2, 7, 7-trimethylquinoline and 4-aryl-7,7-dimethyl-2, 5-dioxo-1, 2, 3, 4, 5, 6, 7, 8-octahydro-quinoline were synthesized by the reaction of aromatic aldehydes, dimedone, ammonium acetate, ethyl acetoacetate or meldrum's acid under microwave irradiation. The reactions were completed with in 2 similar to 8 min giving good yields of 5 or 6.
引用
收藏
页码:313 / 316
页数:4
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