Synthesis and antibacterial activity of oxazolidinone containing sulphonyl group

被引：9
|
作者：
Cui, YJ
Yang, YH [1 ]
Chen, KX
Ji, RY
Zhang, SH
机构：
[1] Chinese Acad Sci, Shanghai Inst Mat Med, Shanghai 200031, Peoples R China
[2] Chinese Acad Sci, Shanghai Inst Biol Sci, Shanghai 200031, Peoples R China
[3] Sichuan Ind Inst Antibiot, Chengdu 610051, Peoples R China
来源：
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2003年 / 13卷 / 14期
关键词：
D O I：
10.1016/S0960-894X(03)00430-X
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A series of oxazolidinone derivatives carrying sulphonyl group was synthesized and their antibacterial activity was evaluated in vitro. Many of such compounds demonstrated potent antibacterial activity. The activity of a novel compound (YC-20) was 2-4-fold more potent than that of linezolid. (C) 2003 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：2311 / 2313
页数：3
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