Synthesis of 2-Substituted Benzothiazoles from 1-Iodo-2-nitrobenzenes by a Copper-Catalyzed One-Pot Three-Component Reaction

被引：18
|
作者：
Liu, Jidan [1 ]
Gui, Qingwen [1 ]
Yang, Zhiyong [1 ]
Tan, Ze [1 ]
Guo, Ruqing [1 ]
Shi, Ji-Cheng [2 ]
机构：
[1] Hunan Univ, State Key Lab Chemo Biosensing & Chemometr, Coll Chem & Chem Engn, Changsha 410082, Hunan, Peoples R China
[2] Guangdong Univ Petrochem Technol, Sch Chem & Life Sci, Maoming 525000, Guangdong, Peoples R China
来源：
SYNTHESIS-STUTTGART | 2013年 / 45卷 / 07期
基金：
美国国家科学基金会;
关键词：
catalysis; copper; multicomponent reactions; heterocycles; cyclizations; sulfur; ONE-STEP SYNTHESIS; S BOND FORMATION; INTRAMOLECULAR CYCLIZATION; SUBSTITUTED BENZOTHIAZOLES; INHIBITORY-ACTIVITY; PARALLEL SYNTHESIS; DNA PHOTOCLEAVAGE; EFFICIENT; 2-ARYLBENZOTHIAZOLES; ANTITUMOR;
D O I：
10.1055/s-0032-1318304
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A novel method was developed for synthesizing 2-substituted 1,3-benzothiazoles through a copper-catalyzed, one-pot, three-component reaction of a 1-iodo-2-nitrobenzene with sodium sulfide and an aldehyde.
引用
收藏
页码：943 / 951
页数：9
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