One-pot three-component reaction providing 1,5-benzodiazepine derivatives

被引：45
|
作者：
Murai, Kenichi [1 ]
Nakatani, Ryo [1 ]
Kita, Yasuyuki [1 ]
Fujioka, Hiromichi [1 ]
机构：
[1] Osaka Univ, Grad Sch Pharmaceut Sci, Suita, Osaka 5650871, Japan
来源：
TETRAHEDRON | 2008年 / 64卷 / 49期
基金：
日本学术振兴会;
关键词：
D O I：
10.1016/j.tet.2008.09.076
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The novel one-pot three-component reaction of aromatic aldehydes, 1,2-phenylenediamine, and beta-keto esters is described. This reaction involves the gamma-selective C-C bond formation of beta-keto esters and produces 1,5-benzodiazepine derivatives. (C) 2008 Elsevier Ltd. All rights reserved.
引用
收藏
页码：11034 / 11040
页数：7
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