N-Arylation of Heterocycles Promoted by Cyclen Derivatives

被引：4
|
作者：
Zhang, Bao-Hua [1 ]
Shi, Lan-xiang [1 ]
Liu, Si-Jie [1 ]
Guo, Rui-Xia [1 ]
机构：
[1] Shijiazhuang Univ, Coll Chem Engn, Shijiazhuang 050035, Peoples R China
来源：
JOURNAL OF HETEROCYCLIC CHEMISTRY | 2015年 / 52卷 / 04期
关键词：
NITROGEN-CONTAINING HETEROCYCLES; COPPER-CATALYZED AMINATION; ARYL HALIDES; C-N; BOND FORMATION; EFFICIENT; LIGAND; AMINES; MILD; AMIDATION;
D O I：
10.1002/jhet.2188
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient copper-catalyzed N-arylation reactions of imidazole, indole, and triazole with aryl or heteroaryl halides using cyclen derivatives as efficient organic base and ligand at moderate temperature have been investigated. The cross-couplings proceed smoothly with good to excellent yields.
引用
收藏
页码：1234 / 1239
页数：6
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