Synthesis and biological evaluation of the first triple inhibitors of human topoisomerase 1, tyrosyl-DNA phosphodiesterase 1 (Tdp1), and tyrosyl-DNA phosphodiesterase 2 (Tdp2)

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作者：
Wang, Ping [1 ]
Elsayed, Mohamed [1 ]
Plescia, Caroline [2 ]
Kiselev, Evgeny [3 ]
Marchand, Christophe [3 ]
Zeleznik, Olga [3 ]
Agama, Keli [3 ]
Pommier, Yves [3 ]
Cushman, Mark [1 ]
机构：
[1] Purdue Univ, MCMP, W Lafayette, IN 47907 USA
[2] Drake Univ, Des Moines, IA 50311 USA
[3] NIH, Bldg 10, Bethesda, MD 20892 USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2017年 / 253卷
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中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
231
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页数：1
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