A concise synthesis of 7-substituted indoles

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作者
Kondo, Y
Kojima, S
Sakamoto, T
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O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
7-Substituted indoles were synthesized by the basic cyclization of 6-substituted tert-butyl 2-(trimethylsilylethynyl)phenylcarbamate which were derived by the lithiation of tert-butyl 2-(trimethylsilylethynyl)phenylcarbamate and the subsequent reaction with electrophiles.
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页码:2741 / 2746
页数:6
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