Discovery of 1,2,3,4-tetrahydrocarbazo-1yl-acetic acids as fatty acid binding protein 4/5 (FABP4/5) inhibitors

被引：0

作者：

Lin, Songnian ^{[1
]}

Deng, Qiaolin ^{[1
]}

Yang, Lihu ^{[1
]}

Chapman, Kevin ^{[1
]}

Wei, Changqing ^{[2
]}

Zhang, Fuzhi ^{[2
]}

Jiao, Zhigang ^{[2
]}

Song, Ji ^{[2
]}

Li, Jinyuan ^{[2
]}

Wu, Hao ^{[2
]}

Qureshi, Sajjad A. ^{[1
]}

Berger, Joel P. ^{[1
]}

Becker, Joe ^{[1
]}

Fitzgerald, Paula ^{[1
]}

Salituro, Gino ^{[1
]}

Sharma, Nandani ^{[1
]}

Xu, Serena ^{[1
]}

Yang, Ruojing ^{[1
]}

Yang, Xiaodong ^{[1
]}

Zhang, Bei B. ^{[1
]}

机构：

[1] Merck Res Labs, Dept Discovery & Preclin Sci, Rahway, NJ 07065 USA

[2] WuXi AppTec, Dept Med Chem, Shanghai 200131, Peoples R China

来源：

ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2012年 / 244卷

关键词：

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

121-MEDI

引用

页数：1

共 50 条

[1] A Critical Role of Fatty Acid Binding Protein 4 and 5 (FABP4/5) in the Systemic Response to Fasting
Syamsunarno, Mas Rizky A. A.
Iso, Tatsuya
Hanaoka, Hirofumi
Yamaguchi, Aiko
Obokata, Masaru
Koitabashi, Norimichi
Goto, Kosaku
Hishiki, Takako
Nagahata, Yoshiko
Matsui, Hiroki
Sano, Motoaki
Kobayashi, Masaki
Kikuchi, Osamu
Sasaki, Tsutomu
Maeda, Kazuhisa
Murakami, Masami
Kitamura, Tadahiro
Suematsu, Makoto
Tsushima, Yoshito
Endo, Keigo
Hotamisligil, Goekhan S.
Kurabayashi, Masahiko
PLOS ONE, 2013, 8 (11):
[2] Discovery of highly selective inhibitors of human fatty acid binding protein 4 (FABP4) by virtual screening
Cai, Haiyan
Yan, Guirui
Zhang, Xiaodong
Gorbenko, Olena
Wang, Heyao
Zhu, Weiliang
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (12) : 3675 - 3679
[3] Small Molecule Inhibitors of Human Adipocyte Fatty Acid Binding Protein (FABP4)
Zhang, Mingming
Zhu, Weiliang
Li, Yingxia
MEDICINAL CHEMISTRY, 2014, 10 (04) : 339 - 347
[4] Role of Fatty Acid Binding Protein 4 (FABP4) in Kidney Disease
Shi, Min
Ma, Liang
Fu, Ping
CURRENT MEDICINAL CHEMISTRY, 2020, 27 (22) : 3657 - 3664
[5] Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review
Floresta, Giuseppe
Pistara, Venerando
Amata, Emanuele
Dichiara, Maria
Marrazzo, Agostino
Prezzavento, Orazio
Rescifina, Antonio
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 138 : 854 - 873
[6] Fatty Acid Binding Protein 4 (FABP4) and the Body Lipid Balance
Kucharski, Miroslaw
Kaczor, Urszula
FOLIA BIOLOGICA-KRAKOW, 2017, 65 (04): : 181 - 186
[7] Fatty acid binding protein 4 (FABP4) and the diagnosis of gestational diabetes
Scifres, Christina
Malczewski, Katie
Catov, Janet
Simhan, Hyagriv
AMERICAN JOURNAL OF OBSTETRICS AND GYNECOLOGY, 2014, 210 (01) : S138 - S138
[8] Identification of new dual FABP4/5 inhibitors based on a naphthalene-1-sulfonamide FABP4 inhibitor
He, Yulong
Dou, Huixia
Gao, Dingding
Wang, Ting
Zhang, Mingming
Wang, Heyao
Li, Yingxia
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 27 (19)
[9] Fatty acid-binding protein 4 (FABP4) and FABP5 modulate cytokine production in the mouse thymic epithelial cells
Adachi, Yasuhiro
Hiramatsu, Sumie
Tokuda, Nobuko
Sharifi, Kazem
Ebrahimi, Majid
Islam, Ariful
Kagawa, Yoshiteru
Vaidyan, Linda Koshy
Sawada, Tomoo
Hamano, Kimikazu
Owada, Yuji
HISTOCHEMISTRY AND CELL BIOLOGY, 2012, 138 (03) : 397 - 406
[10] Fatty acid-binding protein 4 (FABP4) and FABP5 modulate cytokine production in the mouse thymic epithelial cells
Yasuhiro Adachi
Sumie Hiramatsu
Nobuko Tokuda
Kazem Sharifi
Majid Ebrahimi
Ariful Islam
Yoshiteru Kagawa
Linda Koshy Vaidyan
Tomoo Sawada
Kimikazu Hamano
Yuji Owada
Histochemistry and Cell Biology, 2012, 138 : 397 - 406

← 1 2 3 4 5 →