3,5-Dimethylisoxazoles inhibit the bromodomain-histone protein-protein interaction

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作者
Hewings, David S. [1 ,2 ]
Wang, Minghua [2 ]
Philpott, Martin [2 ]
Fedorov, Oleg [2 ]
Uttarkar, Sagar [2 ]
Filippakopoulos, Panagis [2 ]
Picaud, Sarah [2 ]
Vuppusetty, Chaitanya [2 ]
Marsden, Brian [2 ]
Heightman, Tom D. [3 ]
Knapp, Stefan [2 ]
Brennan, Paul [2 ]
Conway, Stuart J. [1 ]
机构
[1] Univ Oxford, Dept Chem, Oxford OX1 3QZ, England
[2] Univ Oxford, Nuffield Dept Clin Med, Struct Genom Consortium, Oxford, England
[3] Astex Pharmaceut, Cambridge, England
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O6 [化学];
学科分类号
0703 ;
摘要
326-MEDI
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页数:1
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