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- [1] Characterization of novel potent and selective anaplastic lymphoma kinase (ALK) inhibitors[J]. JOURNAL OF CLINICAL ONCOLOGY, 2011, 29 (15)Lovly, C. M.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Ingram Canc Ctr, Nashville, TN USAde Stanchina, E.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Ingram Canc Ctr, Nashville, TN USAChen, H.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Ingram Canc Ctr, Nashville, TN USALiang, C.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Ingram Canc Ctr, Nashville, TN USAPao, W.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Ingram Canc Ctr, Nashville, TN USA
- [2] The Discovery and Optimization of a Novel Class of Potent, Selective, and Orally Bioavailable Anaplastic Lymphoma Kinase (ALK) Inhibitors with Potential Utility for the Treatment of Cancer[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (14) : 6523 - 6540Lewis, Richard T.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USABode, Christiane M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAChoquette, Deborah M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAPotashman, Michele论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USARomero, Karina论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAStellwagen, John C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USATeffera, Yohannes论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAMoore, Earl论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAWhittington, Douglas A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAChen, Hao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAEpstein, Linda F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAEmkey, Renee论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAAndrews, Paul S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAYu, Violeta L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USASaffran, Douglas C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAXu, Man论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USADrew, Allison论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USAMerkel, Patricia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USASzilvassy, Steven论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02142 USABrake, Rachael L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02142 USA Amgen Inc, Cambridge, MA 02142 USA
- [3] Anaplastic lymphoma kinase (ALK) inhibitors: a review of design and discovery[J]. MEDCHEMCOMM, 2014, 5 (09) : 1266 - 1279Wang, Wen-Chieh论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, Taiwan Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, TaiwanShiao, Hui-Yi论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, Taiwan Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, TaiwanLee, Chieh-Chien论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, Taiwan Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, TaiwanFung, Ka-Shu论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, Taiwan Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, TaiwanHsieh, Hsing-Pang论文数: 0 引用数: 0 h-index: 0机构: Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, Taiwan Natl Hlth Res Inst, Inst Biotechnol & Pharmaceut Res, Zhunan 35053, Miaoli County, Taiwan
- [4] Discovery of Orally Active Isofuranones as Potent, Selective Inhibitors of Hematopoetic Progenitor Kinase 1[J]. ACS MEDICINAL CHEMISTRY LETTERS, 2021, 12 (03): : 443 - 450Degnan, Andrew P.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAKumi, Godwin K.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAAllard, Christopher W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAAraujo, Erika, V论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAJohnson, Walter L.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Redwood City, CA 94063 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAZimmermann, Kurt论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAPearce, Bradley C.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USASheriff, Steven论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAFutran, Alan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USALi, Xin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USALocke, Gregory A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAYou, Dan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Cambridge, MA 02142 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAMorrison, John论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAParrish, Karen E.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAStromko, Caitlyn论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAMurtaza, Anwar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USALiu, Jinqi论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAJohnson, Benjamin M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Cambridge, MA 02142 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAVite, Gregory D.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAWittman, Mark D.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Cambridge, MA 02142 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA
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- [6] Design and synthesis of a highly selective, orally active and potent anaplastic lymphoma kinase inhibitor (CH5424802)[J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2012, 20 (03) : 1271 - 1280Kinoshita, Kazutomo论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanAsoh, Kohsuke论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanFuruichi, Noriyuki论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanIto, Toshiya论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanKawada, Hatsuo论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanHara, Sousuke论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanOhwada, Jun论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanMiyagi, Takuho论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanKobayashi, Takamitsu论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanTakanashi, Kenji论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanTsukaguchi, Toshiyuki论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanSakamoto, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanTsukuda, Takuo论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanOikawa, Nobuhiro论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan
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