Efficient approach for the parallel solid-phase synthesis of 1,1,3,4-tetrasubstituted-5-oxopiperazin-1-ium compounds

被引：3

作者：

Nefzi, Adel ^{[1
]}

Santos, Rodegar T. ^{[1
]}

机构：

[1] Torrey Pines Inst Mol Studies, San Diego, CA 92121 USA

来源：

TETRAHEDRON LETTERS | 2006年 / 47卷 / 23期

关键词：

D O I：

10.1016/j.tetlet.2006.03.196

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient approach for the design and parallel solid-phase synthesis of unique tetrasubstituted oxopiperazinium derivatives is presented. The synthetic procedure involved a seven-step sequence carried out starting from resin-bound dipeptides. The desired compounds were obtained in good yields and high purity. (c) 2006 Elsevier Ltd. All rights reserved.

引用

页码：3819 / 3822

页数：4

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