Microwave-assisted one step high-throughput synthesis of benzimidazoles

被引：129
|
作者：
Lin, SY [1 ]
Isome, Y [1 ]
Stewart, E [1 ]
Liu, JF [1 ]
Yohannes, D [1 ]
Yu, LB [1 ]
机构：
[1] ArQule Inc, Woburn, MA 01801 USA
来源：
TETRAHEDRON LETTERS | 2006年 / 47卷 / 17期
关键词：
D O I：
10.1016/j.tetlet.2006.02.127
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
One-pot synthesis of benzimidazoles from diamines and carboxylic acids was developed under microwave irradiation condition, which provided a practical and efficient method for high-throughput synthesis of this important class of heterocyclic compounds. (c) 2006 Elsevier Ltd. All rights reserved.
引用
收藏
页码：2883 / 2886
页数：4
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