Palladium-catalyzed reactions on 1,2-diazines

被引:20
|
作者
Maes, BUW
Tapolcsányi, P
Meyers, C
Mátyus, M
机构
[1] Univ Antwerp, Dept Chem, B-2020 Antwerp, Belgium
[2] Semmelweis Univ, Dept Organ Chem, Szentagothai Knowledge Ctr, H-1092 Budapest, Hungary
关键词
D O I
10.2174/138527206775473841
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
In this report, we review the C- and N-functionalization of the pyridazine nucleus via palladium-catalyzed reactions (Suzuki, Stille, Sonogashira, carbonylation, Heck, Buchwald-Hartwig) in which carbon atoms of the pyridazine nucleus are involved. The efficient use of these reactions in synthetic strategies to build up polycyclic 1,2-diazines is also included.
引用
收藏
页码:377 / 417
页数:41
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