Synthesis and evaluation of a new PET ligand for imaging of monoacylglycerol lipase in brain

被引:0
|
作者
Mori, Wakana [1 ]
Kurihara, Yusuke [2 ]
Hatori, Akiko [1 ]
Zhang, Yiding [1 ]
Fujinaga, Masayuki [1 ]
Zhang, Ming-Rong [1 ]
机构
[1] Natl Inst Quantum & Radiol Sci & Technol, Dept Radiopharmaceut Dev, Natl Inst Radiol Sci, Chiba, Japan
[2] SHI Accelerator Serv, Tokyo, Japan
关键词
PRECLINICAL EVALUATION;
D O I
暂无
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
P-238
引用
收藏
页码:S394 / S395
页数:2
相关论文
共 50 条
  • [1] Synthesis and evaluation of PET ligands for monoacylglycerol lipase in brain
    Mori, Wakana
    Kurihara, Yusuke
    Yamasaki, Tomoteru
    Hatori, Akiko
    Fujinaga, Masayuki
    Zhang, Ming-Rong
    NUCLEAR MEDICINE AND BIOLOGY, 2022, 108 : S99 - S99
  • [2] A Novel PET Imaging Probe Targeting Monoacylglycerol Lipase In The Brain
    Wang, Changning
    MULTIPLE SCLEROSIS JOURNAL, 2017, 23 (01) : 64 - 64
  • [3] Development of two new PET radiotracers with different brain kinetics for imaging monoacylglycerol lipase in brain
    Mori, Wakana
    JOURNAL OF NUCLEAR MEDICINE, 2020, 61
  • [4] A novel 18F-labeled reversible PET ligand for imaging monoacylglycerol lipase
    Rong, Jian
    Zhao, Chunyu
    Li, Yinlong
    Chen, Jiahui
    Haider, Ahmed
    Crowe, Ronald
    Collier, Thomas
    Liang, Steven
    NUCLEAR MEDICINE AND BIOLOGY, 2023, 126 : S74 - S74
  • [5] Development of a novel tight-binding reversible PET ligand for imaging monoacylglycerol lipase
    Rong, Jian
    Xia, Xiaotian
    Zhang, Ming-Rong
    Wang, Lu
    Liang, Steven
    JOURNAL OF NUCLEAR MEDICINE, 2021, 62
  • [6] A novel PET ligand for imaging monoacylglycerol lipase in naive and mouse models of Alzheimer's disease
    Rong, Jian
    Chen, Jiahui
    Xia, Xiaotian
    Zhao, Chunyu
    Shao, Tuo
    Xiao Zhiwei
    Pang, Fuwen
    Liang, Steven
    NUCLEAR MEDICINE AND BIOLOGY, 2021, 96-97 : S21 - S21
  • [7] Demonstration of intracellular pH-weighting PET imaging using a new-type PET probe responsible for monoacylglycerol lipase activity in the brain
    Yamasaki, Tomoteru
    Mori, Wakana
    Ohkubo, Takayuki
    Hiraishi, Atsuto
    Kurihara, Yusuke
    Nengaki, Nobuki
    Zhang, Ming-Rong
    NUCLEAR MEDICINE AND BIOLOGY, 2022, 108 : S112 - S113
  • [8] Radiosynthesis and evaluation of novel 18F labeled PET ligands for imaging monoacylglycerol lipase
    Li, Yinlong
    Mori, Wakana
    Chaudhary, Ahmad
    Zhao, Chunyu
    Yamasaki, Tomoteru
    Zhang, Zachary
    Feng, Siyan
    Ware, Tim
    Rong, Jian
    Fujinaga, Masayuki
    Chen, Jiahui
    Kumata, Katsushi
    Zhang, Yiding
    Hu, Kuan
    Xie, Lin
    Zhou, Xin
    Song, Zhendong
    Gao, Yabiao
    Sun, Zhenkun
    Patel, Jimmy S.
    Zhai, Chuangyan
    Yuan, Katherine Y.
    Collier, Thomas L.
    Ran, Chongzhao
    Collin, Ludovic
    Haider, Achi
    Grether, Uwe
    Wittwer, Matthias B.
    Cravatt, Benjamin F.
    Zhang, Ming-Rong
    Liang, Steven H.
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 285
  • [9] In Vitro and in Vivo Evaluation of 11C-Labeled Azetidinecarboxylates for Imaging Monoacylglycerol Lipase by PET Imaging Studies
    Cheng, Ran
    Mori, Wakana
    Ma, Longle
    Alhouayek, Mireille
    Hatori, Akiko
    Zhang, Yiding
    Ogasawara, Daisuke
    Yuan, Gengyang
    Chen, Zhen
    Zhang, Xiaofei
    Shi, Hang
    Yamasaki, Tomoteru
    Xie, Lin
    Kumata, Katsushi
    Fujinaga, Masayuki
    Nagai, Yuji
    Minamimoto, Takafumi
    Svensson, Mona
    Wang, Lu
    Du, Yunfei
    Ondrechen, Mary Jo
    Vasdev, Neil
    Cravatt, Benjamin F.
    Fowler, Christopher
    Zhang, Ming-Rong
    Liang, Steven H.
    JOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (06) : 2278 - 2291
  • [10] Development of reversible monoacylglycerol lipase PET tracers with improved brain uptake
    He, Yingfang
    Schild, Matthias
    Grether, Uwe
    Humm, Roland
    Keller, Claudia
    Schibli, Roger
    Gobbi, Luca
    Mu, Linjing
    NUCLEAR MEDICINE AND BIOLOGY, 2021, 96-97 : S36 - S36