Efficient synthesis and insecticidal activity of novel pyridin-3-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles

被引：0

作者：

Qian, Qun ^{[1
]}

Zhu, Yiwen ^{[1
]}

Zhang, Min ^{[1
]}

Lu, Dongliang ^{[1
]}

Cao, Weiguo ^{[2
]}

Song, Liping ^{[2
]}

Huang, Qingchun ^{[3
]}

机构：

[1] Shanghai Univ, Coll Sci, Dept Chem, Shanghai 200444, Peoples R China

[2] Chinese Acad Sci, Shanghai Inst Organ Chem, Key Lab Organofluorine Chem, Shanghai 200032, Peoples R China

[3] E China Univ Sci & Technol, Sch Pharm, Shanghai Key Lab Chem Biol, Shanghai 200237, Peoples R China

来源：

MONATSHEFTE FUR CHEMIE | 2013年 / 144卷 / 02期

基金：

中国国家自然科学基金;

关键词：

Pyridine; 1,2,4]Triazolo[3,4-b][1,3,4]thiadiazoles; Bioactivity; DERIVATIVES; TRIAZOLE;

D O I：

10.1007/s00706-012-0798-1

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A series of novel [1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles bearing pyridine ring derivatives was synthesized from 2,6-dimethylpyridin-3,5-dicarboxylic acid diethyl ester. The structures of the compounds were characterized by use of IR, NMR, EI-MS, and elemental analysis. The structure of one compound was further confirmed by X-ray diffraction analysis. Biological assays showed that these compounds had potential insecticidal activity with especially strong regulation of the growth of 2nd instar Mythimna separata larvae. The effects on bioactivity of substituent groups on phenyl ring were also screened. .

引用

页码：231 / 236

页数：6

共 50 条

[1] Efficient synthesis and insecticidal activity of novel pyridin-3-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles
Qun Qian
Yiwen Zhu
Min Zhang
Dongliang Lu
Weiguo Cao
Liping Song
Qingchun Huang
Monatshefte für Chemie - Chemical Monthly, 2013, 144 : 231 - 236
[2] Synthesis and antiviral activity of novel [1,2,4]triazolo[3,4b][1,3,4]thiadiazoles, [1,2,4]triazolo[3,4-b][1,3,4]thiadiazines and [1,2,4]triazolo[3,4-b][1,3,4]thiadiazepines
Farghaly, Abdel-Rahman
De Clercq, Erik
El-Kashef, Hussein
ARKIVOC, 2006, : 137 - 151
[3] Efficient Synthesis of Fluorinated [1,2,4]Triazolo[3,4-b][1,3,4]thiadiazoles
B. K. Dhotre
S. V. Raut
V. B. Jagrut
M. A. Patharia
M. A. Pathan
Russian Journal of Organic Chemistry, 2021, 57 : 1135 - 1140
[4] Efficient Synthesis of Fluorinated [1,2,4]Triazolo[3,4-b][1,3,4]thiadiazoles
Dhotre, B. K.
Raut, S. V.
Jagrut, V. B.
Patharia, M. A.
Pathan, M. A.
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, 2021, 57 (07) : 1135 - 1140
[5] Synthesis and Biological Evaluation of Some [1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazoles and [1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazines
Naveena, Channamata Shankara
Poojary, Boja
Chandrashekhar, Chikkanna
Kumari, Nalilu Suchetha
LETTERS IN DRUG DESIGN & DISCOVERY, 2011, 8 (02) : 189 - 200
[6] Synthesis and antimicrobial activities of some new [1,2,4] triazolo[3,4-b][1,3,4]thiadiazoles and [1,2,4]triazolo[3,4-b][1,3,4]thiadiazines
Demirbas, N
Demirbas, A
Karaoglu, SA
Çelik, E
ARKIVOC, 2005, : 75 - 91
[7] Synthesis and Antimicrobial Evaluation of 6-Aryl-3-(pyridin-4-yl)-[1,2,4] triazolo[3,4-b][1,3,4]thiadiazoles
Almehmadi, Mazen
Alsaiari, Ahad Amer
Allahyani, Mamdouh
Aljuaid, Abdulelah
Alsharif, Abdulaziz
Asif, Mohammad
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2023, 33 (02) : 173 - 177
[8] Synthesis of 3-pyridin-4-yl-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazepines
M. V. Karpov
A. V. Khramchikhin
M. D. Stadnichuk
Russian Journal of General Chemistry, 2011, 81
[9] Synthesis of 3-pyridin-4-yl-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazepines
Karpov, M. V.
Khramchikhin, A. V.
Stadnichuk, M. D.
RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2011, 81 (03) : 573 - 575
[10] A CONVENIENT AND NOVEL SYNTHESIS OF 1,2,4-TRIAZOLO[3,4-B][1,3,4]-THIADIAZOLES AS POTENTIAL PESTICIDES
CHATURVEDI, B
TIWARI, N
NIZAMUDDIN
AGRICULTURAL AND BIOLOGICAL CHEMISTRY, 1988, 52 (05): : 1229 - 1232

← 1 2 3 4 5 →