Synthesis and fungicidal activity of new fluorine-containing mandelic acid amide compounds

被引:16
|
作者
Li, Shuai [1 ]
Cui, Can [1 ]
Wang, Man-Yi [1 ]
Yu, Shui-Jing [1 ]
Shi, Yan-Xia [2 ]
Zhang, Xiao [1 ]
Li, Zheng-Ming [1 ]
Zhao, Wei-Guang [1 ]
Li, Bao-Ju [2 ]
机构
[1] Nankai Univ, Natl Pesticide Engn Res Ctr Tianjin, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China
[2] Chinese Acad Agr Sci, Inst Vegetables & Flowers, Beijing 100193, Peoples R China
基金
中国国家自然科学基金;
关键词
Fluorinated mandelic acid amide; Fungicidal activities; Synthesis; DRUGS;
D O I
10.1016/j.jfluchem.2012.02.011
中图分类号
O61 [无机化学];
学科分类号
070301 ; 081704 ;
摘要
A series of novel fluorine-containing mandelic acid amide compounds were designed and synthesized by a facile method, and their structures were characterized by H-1 nuclear magnetic resonance (NMR) and high-resolution mass spectrometry. The preliminary in vivo bioassays indicated that some of the title compounds showed excellent fungicidal activities in vivo against Pseudoperonospora cubensis at the dosage of 25 mg L-1, which were comparable with the control (Mandipropamid). (c) 2012 Elsevier B.V. All rights reserved.
引用
收藏
页码:108 / 112
页数:5
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