Pyrazole Inhibitors of GluN2B NMDA Receptor Subunit

被引：0
|
作者：
Rosse, Gerard [1 ,2 ]
机构：
[1] Dart Neurosci LLC, Struct Guided Chem, 7473 Lusk Blvd, San Diego, CA 92121 USA
[2] Drexel Univ, Coll Med, Dept Physiol & Pharmacol, New Coll Bldg,245 North 15th St, Philadelphia, PA 19102 USA
来源：
ACS MEDICINAL CHEMISTRY LETTERS | 2016年 / 7卷 / 12期
关键词：
D O I：
10.1021/acsmedchemlett.6b00433
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：1018 / 1019
页数：2
相关论文
共 50 条
  • [1] Development of a PET Ligand for Imaging GluN2B Subunit of the NMDA Receptor
    Betzel, Thomas
    Tewes, Bastian
    Frehland, Bastian
    Schepmann, Dirk
    Kraemer, Stefanie D.
    Schibli, Roger
    Wuensch, Bernard
    Ametamey, Simon M.
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2015, 58 : S41 - S41
  • [2] Probing NMDA receptor GluN2A and GluN2B subunit expression and distribution in cortical neurons
    Balsara, Rashna D.
    Ferreira, Ashley N.
    Donahue, Deborah L.
    Castellino, Francis J.
    Sheets, Patrick L.
    NEUROPHARMACOLOGY, 2014, 79 : 542 - 549
  • [3] GluN2B Subunit of the NMDA Receptor: The Keystone of the Effects of Alcohol During Neurodevelopment
    Mickaël Naassila
    Olivier Pierrefiche
    Neurochemical Research, 2019, 44 : 78 - 88
  • [4] GluN2B Subunit of the NMDA Receptor: The Keystone of the Effects of Alcohol During Neurodevelopment
    Naassila, Mickael
    Pierrefiche, Olivier
    NEUROCHEMICAL RESEARCH, 2019, 44 (01) : 78 - 88
  • [5] Memory in aged mice is rescued by enhanced expression of the GluN2B subunit of the NMDA receptor
    Brim, B. L.
    Haskell, R.
    Awedikian, R.
    Ellinwood, N. M.
    Jin, L.
    Kumar, A.
    Foster, T. C.
    Magnusson, K. R.
    BEHAVIOURAL BRAIN RESEARCH, 2013, 238 : 211 - 226
  • [6] Subunit arrangement and phenylethanolamine binding in GluN1/GluN2B NMDA receptors
    Karakas, Erkan
    Simorowski, Noriko
    Furukawa, Hiro
    NATURE, 2011, 475 (7355) : 249 - U170
  • [7] Subunit arrangement and phenylethanolamine binding in GluN1/GluN2B NMDA receptors
    Erkan Karakas
    Noriko Simorowski
    Hiro Furukawa
    Nature, 2011, 475 : 249 - 253
  • [8] GluN2A and GluN2B subunit-containing NMDA receptors in hippocampal plasticity
    Shipton, Olivia A.
    Paulsen, Ole
    PHILOSOPHICAL TRANSACTIONS OF THE ROYAL SOCIETY B-BIOLOGICAL SCIENCES, 2014, 369 (1633)
  • [9] The Apelin/APJ system modulates seizure activity and endocytosis of the NMDA receptor GluN2B subunit
    Zhang, Xiaogang
    Gu, Yixue
    Ma, Yuanlin
    Wu, Junhong
    Chen, Yuanyuan
    Tao, Kaiyan
    Sun, Houchao
    Liu, Zhao
    Wang, Xuefeng
    Tian, Xin
    NEUROCHEMISTRY INTERNATIONAL, 2023, 167
  • [10] Structural basis of subunit selectivity for competitive NMDA receptor antagonists with preference for GluN2A over GluN2B subunits
    Lind, Genevieve E.
    Mou, Tung-Chung
    Tamborini, Lucia
    Pomper, Martin G.
    De Micheli, Carlo
    Conti, Paola
    Pinto, Andrea
    Hansen, Kasper B.
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2017, 114 (33) : E6942 - E6951
12345