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- [1] Discovery and Optimization of C-2 Methyl Imidazopyrrolopyridines as Potent and Orally Bioavailable JAK1 Inhibitors with Selectivity over JAK2[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (13) : 6176 - 6193Zak, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAMendonca, Rohan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABalazs, Mercedesz论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABarrett, Kathy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABergeron, Philippe论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABlair, Wade S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAChang, Christine论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USADeshmukh, Gauri论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USADeVoss, Jason论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USADragovich, Peter S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAEigenbrot, Charles论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGhilardi, Nico论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGibbons, Paul论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGradl, Stefan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHamman, Chris论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHanan, Emily J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHarstad, Eric论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Safety Assessment, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHewitt, Peter R.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHurley, Christopher A.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAJin, Tian论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAJohnson, Adam论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAJohnson, Tony论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKenny, Jane R.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKoehler, Michael F. T.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKohli, Pawan Bir论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKulagowski, Janusz J.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALabadie, Sharada论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALiao, Jiangpeng论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALiimatta, Marya论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALin, Zhonghua论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALupardus, Patrick J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAMaxey, Robert J.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAMurray, Jeremy M.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAPulk, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USARodriguez, Madeleine论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USASavage, Scott论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Small Mol Proc Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAShia, Steven论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USASteffek, Micah论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAUbhayakar, Savita论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAUltsch, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAvan Abbema, Anne论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAWard, Stuart I.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAXiao, Ling论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAXiao, Yisong论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA
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