Discovery and optimization of potent, selective, and orally bioavailable Jak1 inhibitors

被引:0
|
作者
Zak, Mark [1 ]
Johnson, Adam [1 ]
Van Abbema, Anne [1 ]
Waszkowycz, Bohdan [2 ]
Eigenbrot, Charles [1 ]
Chang, Christine [1 ]
Hurley, Christopher [2 ]
Hanan, Emily [1 ]
Kenny, Jane [1 ]
Kulagowski, Janusz [2 ]
DeVoss, Jason [1 ]
Murray, Jeremy [1 ]
Balazs, Mercedesz [1 ]
Steffek, Micah [1 ]
Koehler, Michael [1 ]
Ghilardi, Nico [1 ]
Chakravarty, Paroma [1 ]
Lupardus, Patrick [1 ]
Gibbons, Paul [1 ]
Dragovich, Peter [1 ]
Bergeron, Philippe [1 ]
Pulk, Rebecca [1 ]
Mendonca, Rohan [1 ]
Savage, Scott [1 ]
Labadie, Sharada [1 ]
Gradl, Stefan [1 ]
Ward, Stuart [2 ]
Blair, Wade [1 ]
Jia, Wei [1 ]
机构
[1] Genentech Inc, San Francisco, CA 94080 USA
[2] Argenta, Harlow CM19 5TR, Essex, England
关键词
D O I
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
259-MEDI
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收藏
页数:1
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