Pyridazines .84. Pyridazino[3,4-e]pyrido[3,2-b][1,4]diazepine, a novel tricyclic ring system

被引：6
|
作者：
Heinisch, G
Matuszczak, B
机构：
[1] Inst. of Pharmaceutical Chemistry, University of Innsbruck, A-6020 Innsbruck
来源：
JOURNAL OF HETEROCYCLIC CHEMISTRY | 1997年 / 34卷 / 05期
关键词：
D O I：
10.1002/jhet.5570340508
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The preparation of pyridazino[3,4-e]pyrido[3,2-b][1,4]diazepin-5-ones 8 and 9 starting from appropriately substituted pyridazine-4-carboxamides is reported. The new compounds were tested for HIV-1 reverse transcriptase inhibitory activity.
引用
收藏
页码：1421 / 1425
页数：5
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