The synthesis of substituted phenylpyrimidines via Suzuki coupling reactions

被引：28

作者：

Delia, TJ ^{[1
]}

Schomaker, JM ^{[1
]}

Kalinda, AS ^{[1
]}

机构：

[1] Cent Michigan Univ, Dept Chem, Malcolm H Filson Labs, Mt Pleasant, MI 48859 USA

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2006年 / 43卷 / 01期

关键词：

D O I：

10.1002/jhet.5570430119

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

This paper describes the mon-, di-, and triarylation of the pyrimidine ring. It is possible to introduce one or more aryl rings in generally good yields and in a specific order, namely first in position 4, second in position 6, followed by position 2. A study of solvent and catalyst requirements has also been conducted.

引用

页码：127 / 131

页数：5

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