SLOW AND FAST INACTIVATION OF HNAV1.3 VOLTAGE-GATED SODIUM CHANNELS BY ESLICARBAZEPINE, R-LICARBAZEPINE AND LACOSAMIDE

被引:0
|
作者
Soares-da-Silva, P. [1 ,2 ]
Hebeisen, S. [3 ]
机构
[1] Bial Portela & Ca SA, Trofa, Portugal
[2] Univ Porto, P-4100 Oporto, Portugal
[3] BSYS GmbH, Witterswil, Switzerland
关键词
D O I
暂无
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
引用
收藏
页码:152 / 152
页数:1
相关论文
共 50 条
  • [1] Slow and fast inactivation of hNav1.3 voltage-gated sodium channels by eslicarbazepine, R-licarbazepine and lacosamide
    Soares-da-Silva, P.
    Heibesen, S.
    JOURNAL OF NEUROLOGY, 2013, 260 : S196 - S197
  • [2] Slow and fast inactivation of hNav1.3 voltage-gated sodium channels by eslicarbazepine, oxcarbazepine and carbamazepine
    Heibesen, S.
    Soares-da-Silva, P.
    JOURNAL OF NEUROLOGY, 2013, 260 : S30 - S30
  • [3] SLOW AND FAST INACTIVATION OF HNAV1.3 VOLTAGE-GATED SODIUM CHANNELS BY ESLICARBAZEPINE, OXCARBAZEPINE AND CARBAMAZEPINE
    Hebeisen, S.
    Soares-da-Silva, P.
    EPILEPSIA, 2013, 54 : 152 - 152
  • [4] EFFECTS OF ESLICARBAZEPINE, R-LICARBAZEPINE AND OXCARBAZEPINE ON FAST AND SLOW INACTIVATION OF VOLTAGE-GATED SODIUM CHANNELS
    Aires, C.
    Hebeisen, S.
    Soares-Da-Silva, P.
    EPILEPSIA, 2012, 53 : 51 - 51
  • [5] EFFECTS OF ESLICARBAZEPINE AND LACOSAMIDE ON SLOW AND FAST INACTIVATION OF VOLTAGE-GATED SODIUM CHANNELS
    Bonifacio, M. J.
    Hebeisen, S.
    Soares-Da-Silva, P.
    EPILEPSIA, 2012, 53 : 124 - 124
  • [6] SLOW AND FAST INACTIVATION OF VOLTAGE-GATED SODIUM CHANNELS BY ESLICARBAZEPINE AND CARBAMAZEPINE
    Soares-Da-Silva, P.
    Hebeisen, S.
    EPILEPSIA, 2012, 53 : 54 - 54
  • [7] Eslicarbazepine and the enhancement of slow inactivation of voltage-gated sodium channels: A comparison with carbamazepine, oxcarbazepine and lacosamide
    Hebeisen, Simon
    Pires, Nuno
    Loureiro, Ana I.
    Bonifacio, Maria Joao
    Palma, Nuno
    Whyment, Andrew
    Spanswick, David
    Soares-da-Silva, Patricio
    NEUROPHARMACOLOGY, 2015, 89 : 122 - 135
  • [8] THE EFFECTS OF ESLICARBAZEPINE, R-LICARBAZEPINE, OXCARBAZEPINE AND CARBAMAZEPINE ON SODIUM CURRENTS THROUGH NAV1.3 CHANNELS
    Wright, L.
    Brady, K.
    Hebeisen, S.
    Soares-Da-Silva, P.
    EPILEPSIA, 2012, 53 : 197 - 197
  • [9] The Investigational anticonvulsant lacosamide selectively enhances slow inactivation of voltage-gated sodium channels
    Errington, Adam C.
    Stoehr, Thomas
    Heers, Cara
    Lees, George
    MOLECULAR PHARMACOLOGY, 2008, 73 (01) : 157 - 169
  • [10] Accessibility of the fast inactivation gate is independent of slow inactivation for voltage-gated sodium channels.
    Vedantham, V
    Cannon, SC
    BIOPHYSICAL JOURNAL, 1998, 74 (02) : A31 - A31