Stimulation of G-protein Gαi3 subunits by h5-HT1A receptors expressed in CHO cells:: Agonists concentration-response curves

被引:0
|
作者
Newman-Tancredi, A [1 ]
Cussac, D [1 ]
Marini, L [1 ]
Millan, MJ [1 ]
机构
[1] Inst Rech Servier, Dept Psychopharmacol, F-78290 Croissy Sur Seine, France
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
188P
引用
收藏
页数:1
相关论文
共 36 条
  • [1] G-protein activation by H5-HT1B receptors expressed in CHO cells:: Acintillation proximity assays reveal constitutive Gaαi3 activation.
    Newman-Tancredi, A
    Cussac, D
    Touzard, M
    Chaput, C
    Marini, L
    Millan, MJ
    BRITISH JOURNAL OF PHARMACOLOGY, 2002, 135
  • [2] Antibody capture assay reveals bell-shaped concentration-response isotherms for h5-HT1A receptor-mediated Gαi3 activation:: Conformational selection by high-efficacy agonists, and relationship to trafficking of receptor signaling
    Newman-Tancredi, A
    Cussac, D
    Marini, L
    Millan, MJ
    MOLECULAR PHARMACOLOGY, 2002, 62 (03) : 590 - 601
  • [3] Suppression of cellular invasion by activated G-protein subunits Gαo, Gαi1, Gαi2, and Gαi3 and sequestration of Gβγ
    Faivre, S
    Régnauld, K
    Bruyneel, E
    Nguyen, QD
    Mareel, M
    Emami, S
    Gespach, C
    MOLECULAR PHARMACOLOGY, 2001, 60 (02) : 363 - 372
  • [4] Competitive interaction of 5-HT1A receptors with G-protein subtypes in CHO cells demonstrated by RNA interference
    Rauly-Lestienne, Isabelle
    Lestienne, Fabrice
    Ailhaud, Marie-Christine
    Binesse, Johan
    Newman-Tancredi, Adrian
    Cussac, Didier
    CELLULAR SIGNALLING, 2011, 23 (01) : 58 - 64
  • [5] Differential ligand efficacy at h5-HT1A receptor-coupled G-protein subtypes:: a commentary
    Newman-Tancredi, A
    INVERSE AGONISM, 2003, 1249 : 101 - 117
  • [6] HUMAN 5-HT1A RECEPTOR EXPRESSED IN INSECT CELLS ACTIVATES ENDOGENOUS G(O)-LIKE G-PROTEIN(S)
    MULHERON, JG
    CASANAS, SJ
    ARTHUR, JM
    GARNOVSKAYA, MN
    GETTYS, TW
    RAYMOND, JR
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1994, 269 (17) : 12954 - 12962
  • [7] SELECTIVE ACTIVATION OF INHIBITORY G-PROTEIN ALPHA-SUBUNITS BY PARTIAL AGONISTS OF THE HUMAN 5-HT(1A) RECEPTOR
    GETTYS, TW
    FIELDS, TA
    RAYMOND, JR
    BIOCHEMISTRY, 1994, 33 (14) : 4283 - 4290
  • [8] Estimation of 'full' inverse agonism at G-protein-coupled receptors by [35S]-GTPγS binding at h5-HT1D receptors expressed in CHO cells
    Audinot, V
    Newman-Tancredi, A
    Millan, MJ
    BRITISH JOURNAL OF PHARMACOLOGY, 1999, 126 : U47 - U47
  • [9] 5-HT1A receptor activates Na+/H+ exchange in CHO-K1 cells through G(i alpha 2) and G(i alpha 3)
    Garnovskaya, MN
    Gettys, TW
    vanBiesen, T
    Prpic, V
    Chuprun, JK
    Raymond, JR
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1997, 272 (12) : 7770 - 7776
  • [10] DIFFERENT EFFICIENCY OF G-PROTEIN COUPLING OF THE RAT D-2L AND D-3 DOPAMINE-RECEPTORS EXPRESSED IN CHO CELLS
    GARDNER, B
    HALL, DA
    STRANGE, PG
    BRITISH JOURNAL OF PHARMACOLOGY, 1995, 115 : P104 - P104