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- [1] A Phase 1 study of ARQ 087, an oral pan-FGFR inhibitor in patients with advanced solid tumoursBRITISH JOURNAL OF CANCER, 2017, 117 (11) : 1592 - 1599Papadopoulos, K. P.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USAEl-Rayes, B. F.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, 1365-C Clifton Rd NE, Atlanta, GA 30322 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USATolcher, A. W.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USAPatnaik, A.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USARasco, D. W.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USAHarvey, R. D.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, 1365-C Clifton Rd NE, Atlanta, GA 30322 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USALoRusso, P. M.论文数: 0 引用数: 0 h-index: 0机构: Karmanos Canc Inst, 4206-4th Floor HWCRC,4100 John R, Detroit, MI 48201 USA Yale Univ, Canc Ctr, 55 Pk St,Ste First Floor, New Haven, CT 06519 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USASachdev, J. C.论文数: 0 引用数: 0 h-index: 0机构: Scottsdale Healthcare, Virginia G Piper Canc Ctr, 10460N 92nd St, Scottsdale, AZ 85258 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USAAbbadessa, G.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, One Wall St, Burlington, MA 01803 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USASavage, R. E.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, One Wall St, Burlington, MA 01803 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USAHall, T.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, One Wall St, Burlington, MA 01803 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USASchwartz, B.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, One Wall St, Burlington, MA 01803 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USAWang, Y.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, One Wall St, Burlington, MA 01803 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USAKazakin, J.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, One Wall St, Burlington, MA 01803 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USAShaib, W. L.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, 1365-C Clifton Rd NE, Atlanta, GA 30322 USA South Texas Accelerated Res Therapeut, 4383 Med Dr, San Antonio, TX 78229 USA
- [2] A Phase 1 study of ARQ 087, an oral pan-FGFR inhibitor in patients with advanced solid tumoursBritish Journal of Cancer, 2017, 117 : 1592 - 1599K P Papadopoulos论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,B F El-Rayes论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,A W Tolcher论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,A Patnaik论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,D W Rasco论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,R D Harvey论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,P M LoRusso论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,J C Sachdev论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,G Abbadessa论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,R E Savage论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,T Hall论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,B Schwartz论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,Y Wang论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,J Kazakin论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,W L Shaib论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Research Therapeutics,
- [3] A phase 1, dose-escalation, first-in-human study of ARQ 087, an oral pan-FGFR inhibitor, in adult subjects with advanced solid tumorsEUROPEAN JOURNAL OF CANCER, 2014, 50 : 125 - 125Papadopoulos, K.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USATolcher, A.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USAKittaneh, M.论文数: 0 引用数: 0 h-index: 0机构: Karmanos Canc Inst, Ctr Translat Therapeut, Detroit, MI USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USAPatniak, A.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USARasco, D.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USAChambers, G.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USANewth, G.论文数: 0 引用数: 0 h-index: 0机构: Karmanos Canc Inst, Ctr Translat Therapeut, Detroit, MI USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USASavage, R.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Clin Dev, Woburn, MA USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USAHall, T.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Clin Dev, Woburn, MA USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USASchwartz, B.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Clin Dev, Woburn, MA USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USAKazakin, J.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Clin Dev, Woburn, MA USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USALoRusso, P.论文数: 0 引用数: 0 h-index: 0机构: Karmanos Canc Inst, Ctr Translat Therapeut, Detroit, MI USA South Texas Accelerated Res Therapeut, Med Oncol, San Antonio, TX USA
- [4] ARQ 087, an oral pan- fibroblast growth factor receptor (FGFR) inhibitor, in patients (pts) with advanced and/or metastatic intrahepatic cholangiocarcinoma (iCCA)ANNALS OF ONCOLOGY, 2016, 27 : 109 - 109Mazzaferro, V.论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Inst, Ist Nazl Tumori, Milan, Italy Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyShaib, W.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Sch Med, Winship Canc Inst, Atlanta, GA USA Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyRimassa, L.论文数: 0 引用数: 0 h-index: 0机构: Ist Clin Humanitas IRCCS, Humanitas Canc Ctr, Rozzano, Italy Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyHarris, W.论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Sch Med, Seattle, WA USA Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyPersoneni, N.论文数: 0 引用数: 0 h-index: 0机构: Ist Clin Humanitas IRCCS, Humanitas Canc Ctr, Rozzano, Italy Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyEl-Rayes, B.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Sch Med, Winship Canc Inst, Atlanta, GA USA Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyTolcher, A.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, San Antonio, TX USA Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyHall, T.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Burlington, MA USA Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyWang, Y.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Burlington, MA USA Natl Canc Inst, Ist Nazl Tumori, Milan, ItalySchwartz, B.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Woburn, MA USA Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyKazakin, J.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Burlington, MA USA Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyBusset, M. Droz Dit论文数: 0 引用数: 0 h-index: 0机构: Ist Nazl Tumori, Milan, Italy Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyCotsoglou, C.论文数: 0 引用数: 0 h-index: 0机构: Ist Nazl Tumori, Milan, Italy Natl Canc Inst, Ist Nazl Tumori, Milan, ItalyPapadopoulos, K.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, San Antonio, TX USA Natl Canc Inst, Ist Nazl Tumori, Milan, Italy
- [5] ARQ 087, an oral pan-fibroblast growth factor receptor (FGFR) inhibitor, in patients (pts) with advanced intrahepatic cholangiocarcinoma (iCCA) with FGFR2 genetic aberrations.JOURNAL OF CLINICAL ONCOLOGY, 2017, 35Mazzaferro, Vincenzo论文数: 0 引用数: 0 h-index: 0El-Rayes, Bassel F.论文数: 0 引用数: 0 h-index: 0Cotsoglou, Christian论文数: 0 引用数: 0 h-index: 0Harris, William Proctor论文数: 0 引用数: 0 h-index: 0Damjanov, Nevena论文数: 0 引用数: 0 h-index: 0Masi, Gianluca论文数: 0 引用数: 0 h-index: 0Rimassa, Lorenza论文数: 0 引用数: 0 h-index: 0Personeni, Nicola论文数: 0 引用数: 0 h-index: 0Braiteh, Fadi S.论文数: 0 引用数: 0 h-index: 0Zagonel, Vittorina论文数: 0 引用数: 0 h-index: 0Papadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0Hall, Terence论文数: 0 引用数: 0 h-index: 0Wang, Yunxia论文数: 0 引用数: 0 h-index: 0Abbadessa, Giovanni论文数: 0 引用数: 0 h-index: 0Schwartz, Brian E.论文数: 0 引用数: 0 h-index: 0Kazakin, Julia论文数: 0 引用数: 0 h-index: 0Busset, Michele Droz Dit论文数: 0 引用数: 0 h-index: 0Shaib, Walid La Bib论文数: 0 引用数: 0 h-index: 0
- [6] Phase 1, first-in-human study of ARQ 087, an oral pan-Fibroblast Growth Factor Receptor (FGFR) inhibitor, in patients (pts) with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2015, 33 (15)Papadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USATolcher, Anthony W.论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USAPatnaik, Amita论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USARasco, Drew Warren论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USAChambers, Glenda论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USABeeram, Murali论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USASavage, Ronald论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USAHall, Terence论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USASchwartz, Brian E.论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USAKazakin, Julia论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USALoRusso, Patricia论文数: 0 引用数: 0 h-index: 0机构: START Ctr Canc Care, San Antonio, TX USA
- [7] Phase I study of BGJ398, a selective pan-FGFR inhibitor in genetically preselected advanced solid tumorsCANCER RESEARCH, 2014, 74 (19)Sequist, Lecia V.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA 02114 USA Massachusetts Gen Hosp, Boston, MA 02114 USACassier, Phillippe论文数: 0 引用数: 0 h-index: 0机构: Ctr Leon Berard, F-69373 Lyon, France Massachusetts Gen Hosp, Boston, MA 02114 USAVarga, Andrea论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, France Massachusetts Gen Hosp, Boston, MA 02114 USATabernero, Josep论文数: 0 引用数: 0 h-index: 0机构: Vall dHebron Univ Hosp, Barcelona, Spain Massachusetts Gen Hosp, Boston, MA 02114 USASchellens, Jan H.论文数: 0 引用数: 0 h-index: 0机构: Netherlands Canc Inst, Amsterdam, Netherlands Massachusetts Gen Hosp, Boston, MA 02114 USADelord, Jean-Pierre论文数: 0 引用数: 0 h-index: 0机构: Inst Claudius Regaud, Toulouse, France Massachusetts Gen Hosp, Boston, MA 02114 USALoRusso, Patricia论文数: 0 引用数: 0 h-index: 0机构: Karmanos Canc Inst, Detroit, MI USA Massachusetts Gen Hosp, Boston, MA 02114 USACamidge, D. Ross论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Aurora, CO USA Massachusetts Gen Hosp, Boston, MA 02114 USAHidalgo Medina, Manuel论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Madrid, Spain Massachusetts Gen Hosp, Boston, MA 02114 USASchuler, Martin论文数: 0 引用数: 0 h-index: 0机构: Univ Duisburg Essen, West German Canc Ctr, Essen, Germany Massachusetts Gen Hosp, Boston, MA 02114 USACampone, Mario论文数: 0 引用数: 0 h-index: 0机构: Ctr Rene Gauducheau, F-44035 Nantes, France Massachusetts Gen Hosp, Boston, MA 02114 USATian, G. Gary论文数: 0 引用数: 0 h-index: 0机构: West Clin, Memphis, TN USA Massachusetts Gen Hosp, Boston, MA 02114 USAWong, Steven论文数: 0 引用数: 0 h-index: 0机构: UCLA Med Ctr, Los Angeles, CA USA Massachusetts Gen Hosp, Boston, MA 02114 USACorral, Jesus论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Virgen del Rocio, Seville, Spain Massachusetts Gen Hosp, Boston, MA 02114 USAIsaacs, Randi论文数: 0 引用数: 0 h-index: 0机构: Novartis OTM, E Hanover, NJ USA Massachusetts Gen Hosp, Boston, MA 02114 USASen, Suman K.论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Massachusetts Gen Hosp, Boston, MA 02114 USAPorta, Diana Graus论文数: 0 引用数: 0 h-index: 0机构: NIBR Oncol, Basel, Switzerland Massachusetts Gen Hosp, Boston, MA 02114 USAKulkarni, Swarupa G.论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Massachusetts Gen Hosp, Boston, MA 02114 USALefebvre, Caroline论文数: 0 引用数: 0 h-index: 0机构: Novartis OTM, Basel, Switzerland Massachusetts Gen Hosp, Boston, MA 02114 USAWolf, Juergen论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Cologne, Cologne, Germany Massachusetts Gen Hosp, Boston, MA 02114 USA
- [8] Safety and efficacy of the pan-FGFR inhibitor erdafitinib in advanced urothelial carcinoma and other solid tumors: A systematic review and meta-analysisFRONTIERS IN ONCOLOGY, 2023, 12Zheng, Xinyi论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R China Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R ChinaWang, Hang论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R China Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R ChinaDeng, Junyue论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, West China Hosp, Dept Biotherapy, Chengdu, Sichuan, Peoples R China Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R ChinaYao, Minghe论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R China Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R ChinaZou, Xiuhe论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, West China Hosp, Dept Thyroid Surg, Chengdu, Sichuan, Peoples R China Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R ChinaZhang, Fan论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, West China Hosp, Hlth Management Ctr, Gen Practice Ctr, Chengdu, Peoples R China Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R ChinaMa, Xuelei论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, West China Hosp, Dept Biotherapy, Chengdu, Sichuan, Peoples R China Sichuan Univ, West China Sch Med, Chengdu, Sichuan, Peoples R China
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