共 25 条
- [1] WD Repeat-containing Protein 5 (WDR5) Localizes to the Midbody and Regulates AbscissionJOURNAL OF BIOLOGICAL CHEMISTRY, 2015, 290 (14) : 8987 - 9001Bailey, Jeffrey K.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USAFields, Alexander T.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USACheng, Kaijian论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USALee, Albert论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USAWagenaar, Eric论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USALagrois, Remy论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USASchmidt, Bailey论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USAXia, Bin论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USAMa, Dzwokai论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Neurosci Res Inst, Santa Barbara, CA 93106 USA
- [2] Targeting WD Repeat-Containing Protein 5 (WDR5): A Medicinal Chemistry PerspectiveJOURNAL OF MEDICINAL CHEMISTRY, 2021, 64 (15) : 10537 - 10556Chen, Xin论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R ChinaXu, Junjie论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R ChinaWang, Xianghan论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R ChinaLong, Guanlu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R ChinaYou, Qidong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R ChinaGuo, Xiaoke论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Sch Pharm, Nanjing 210009, Peoples R China
- [3] Upon Infection, Cellular WD Repeat-Containing Protein 5 (WDR5) Localizes to Cytoplasmic Inclusion Bodies and Enhances Measles Virus ReplicationJOURNAL OF VIROLOGY, 2018, 92 (05)Ma, Dzwokai论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USAGeorge, Cyril X.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USANomburg, Jason L.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Harvard Med Sch, Virol Program, Boston, MA USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USAPfaller, Christian K.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Mol Med, Rochester, MN USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USACattaneo, Roberto论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Mol Med, Rochester, MN USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USASamuel, Charles E.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA Univ Calif Santa Barbara, Dept Mol Cellular & Dev Biol, Santa Barbara, CA 93106 USA
- [4] Discovery and Structure-Based Design of Inhibitors of the WD Repeat-Containing Protein 5 (WDR5)-MYC InteractionJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (12) : 8310 - 8323Ding, Jian论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USALiu, Lulu论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAChiang, Ying-Ling论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, Cambridge, MA 02139 USAZhao, Mengxi论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, Cambridge, MA 02139 USALiu, Hejun论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, San Diego, CA 92121 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAYang, Fei论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAShen, Lingling论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USALin, Ying论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, Cambridge, MA 02139 USADeng, Huiwen论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, Cambridge, MA 02139 USAGao, Jingyan论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, Cambridge, MA 02139 USASage, David R.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAWest, Laura论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USALlamas, Luis A.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAHao, Xin论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, Cambridge, MA 02139 USAKawatkar, Sameer论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USALi, En论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, Cambridge, MA 02139 USAJain, Rishi K.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USATallarico, John A.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USACanham, Stephen M.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAWang, He论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, Cambridge, MA 02139 USA
- [5] Design, Synthesis, and Evaluation of WD-Repeat-Containing Protein 5 (WDR5) DegradersJOURNAL OF MEDICINAL CHEMISTRY, 2021, 64 (15) : 10682 - 10710Doelle, Anja论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyAdhikari, Bikash论文数: 0 引用数: 0 h-index: 0机构: Univ Wurzburg, Theodor Boveri Inst, Canc Syst Biol Grp, D-97074 Wurzburg, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyKraemer, Andreas论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Inst Pharmazeut Chem, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany论文数: 引用数: h-index:机构:Berner, Nicola论文数: 0 引用数: 0 h-index: 0机构: Tech Univ Munich, Chair Prote & Bioanalyt, D-85354 Freising Weihenstephan, Germany German Canc Res Ctr, German Canc Consortium DKTK, D-69120 Heidelberg, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyBerger, Lena-Marie论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Inst Pharmazeut Chem, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany论文数: 引用数: h-index:机构:Szewczyk, Magdalena M.论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany论文数: 引用数: h-index:机构:Arrowsmith, Cheryl H.论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Toronto, ON M5G 2C1, Canada Univ Toronto, Dept Med Biophys, Toronto, ON M5G 2M9, Canada Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyGebel, Jakob论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Inst Biophys Chem, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Ctr Biomol Magnet Resonance, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Cluster Excellence Macromol Complexes CEF, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyLoehr, Frank论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Inst Biophys Chem, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Ctr Biomol Magnet Resonance, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Cluster Excellence Macromol Complexes CEF, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyDoetsch, Volker论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany Univ Toronto, Dept Med Biophys, Toronto, ON M5G 2M9, Canada Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyEilers, Martin论文数: 0 引用数: 0 h-index: 0机构: Univ Wurzburg, Theodor Boveri Inst, Dept Biochem & Mol Biol, D-97074 Wurzburg, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyHeinzlmeir, Stephanie论文数: 0 引用数: 0 h-index: 0机构: Tech Univ Munich, Chair Prote & Bioanalyt, D-85354 Freising Weihenstephan, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyKuster, Bernhard论文数: 0 引用数: 0 h-index: 0机构: Tech Univ Munich, Chair Prote & Bioanalyt, D-85354 Freising Weihenstephan, Germany German Canc Res Ctr, German Canc Consortium DKTK, D-69120 Heidelberg, Germany Tech Univ Munich, Bavarian Biomol Mass Spectrometry Ctr BayBioMS, D-85354 Freising Weihenstephan, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanySotriffer, Christoph论文数: 0 引用数: 0 h-index: 0机构: Univ Wurzburg, Inst Pharm & Lebensmittelchem, D-97074 Wurzburg, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyWolf, Elmar论文数: 0 引用数: 0 h-index: 0机构: Univ Warzburg, Theodor Boveri Inst, Canc Syst Biol Grp, D-97074 Wurzburg, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, GermanyKnapp, Stefan论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany Goethe Univ Frankfurt Main, Inst Pharmazeut Chem, D-60438 Frankfurt, Germany German Canc Res Ctr, German Canc Consortium DKTK, D-69120 Heidelberg, Germany Goethe Univ Frankfurt Main, Buchmann Inst Life Sci BMLS, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany
- [6] Discovery of WD Repeat-Containing Protein 5 (WDR5)-MYC Inhibitors Using Fragment-Based Methods and Structure-Based DesignJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (08) : 4315 - 4333Simon, Selena Chacon论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAWang, Feng论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAThomas, Lance R.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Cell & Dev Biol, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAPhan, Jason论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAZhao, Bin论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAOlejniczak, Edward T.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAMacdonald, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAShaw, J. Grace论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USASchlund, Caden论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAPayne, William论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USACreighton, Joy论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Cell & Dev Biol, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAStauffer, Shaun R.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Dept Chem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAWaterson, Alex G.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Dept Chem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USATansey, William P.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Cell & Dev Biol, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USAFesik, Stephen W.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Dept Chem, Nashville, TN 37232 USA Vanderbilt Univ, Sch Med, Dept Biochem, Nashville, TN 37232 USA
- [7] Recent Progress in Modulation of WD40-Repeat Domain 5 Protein (WDR5): Inhibitors and DegradersCANCERS, 2023, 15 (15)Gurung, Raju论文数: 0 引用数: 0 h-index: 0机构: Gachon Univ, Coll Pharm, 191 Hambakmoe Ro, Incheon 21936, South Korea Gachon Univ, Coll Pharm, 191 Hambakmoe Ro, Incheon 21936, South KoreaOm, Darlami论文数: 0 引用数: 0 h-index: 0机构: Gachon Univ, Coll Pharm, 191 Hambakmoe Ro, Incheon 21936, South Korea Gachon Univ, Coll Pharm, 191 Hambakmoe Ro, Incheon 21936, South KoreaPun, Rabin论文数: 0 引用数: 0 h-index: 0机构: Gachon Univ, Coll Pharm, 191 Hambakmoe Ro, Incheon 21936, South Korea Gachon Univ, Coll Pharm, 191 Hambakmoe Ro, Incheon 21936, South Korea论文数: 引用数: h-index:机构:Shin, Dongyun论文数: 0 引用数: 0 h-index: 0机构: Gachon Univ, Coll Pharm, 191 Hambakmoe Ro, Incheon 21936, South Korea Gachon Univ, Gachon Inst Pharmaceut Sci, 191 Hambakmoe Ro, Incheon 21936, South Korea Gachon Univ, Coll Pharm, 191 Hambakmoe Ro, Incheon 21936, South Korea
- [8] The WD repeat-containing protein 5 (WDR5) antagonist WDR5-0103 restores the efficacy of cytotoxic drugs in multidrug-resistant cancer cells overexpressing ABCB1 or ABCG2BIOMEDICINE & PHARMACOTHERAPY, 2022, 154论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Tseng, Han-Yu论文数: 0 引用数: 0 h-index: 0机构: Chang Gung Univ, Coll Med, Grad Inst Biomed Sci, Taoyuan, Taiwan Chang Gung Univ, Coll Med, Grad Inst Biomed Sci, Taoyuan, TaiwanHuang, Yang-Hui论文数: 0 引用数: 0 h-index: 0机构: Chang Gung Univ, Coll Med, Grad Inst Biomed Sci, Taoyuan, Taiwan Chang Gung Univ, Coll Med, Grad Inst Biomed Sci, Taoyuan, TaiwanLi, Yan-Qing论文数: 0 引用数: 0 h-index: 0机构: Chang Gung Univ, Coll Med, Grad Inst Biomed Sci, Taoyuan, Taiwan Chang Gung Univ, Coll Med, Grad Inst Biomed Sci, Taoyuan, TaiwanHung, Tai-Ho论文数: 0 引用数: 0 h-index: 0机构: Taipei Chang Gung Mem Hosp, Dept Obstet & Gynecol, Taipei, Taiwan Chang Gung Univ, Coll Med, Dept Med, Taoyuan, Taiwan Keelung Chang Gung Mem Hosp, Dept Obstet & Gynecol, Keelung, Taiwan Chang Gung Univ, Coll Med, Grad Inst Biomed Sci, Taoyuan, TaiwanWang, Shun-Ping论文数: 0 引用数: 0 h-index: 0机构: Taichung Vet Gen Hosp, Dept Orthoped, Taichung, Taiwan Chang Gung Univ, Coll Med, Grad Inst Biomed Sci, Taoyuan, TaiwanWu, Yu-Shan论文数: 0 引用数: 0 h-index: 0机构: Tunghai Univ, Dept Chem, 181 Taichung Harbor Rd Sect 3, Taichung, Taiwan Chang Gung Univ, Coll Med, Grad Inst Biomed Sci, Taoyuan, Taiwan
- [9] Structure-Based Optimization of a Small Molecule Antagonist of the Interaction Between WD Repeat-Containing Protein 5 (WDR5) and Mixed-Lineage Leukemia 1 (MLL1)JOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (06) : 2478 - 2496Getlik, Matthaeus论文数: 0 引用数: 0 h-index: 0机构: Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, Canada Merck KGaA, Performance Mat, Frankfurter Str 250, D-64289 Darmstadt, Germany Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaSmil, David论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaZepeda-Velazquez, Carlos论文数: 0 引用数: 0 h-index: 0机构: Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaBolshan, Yuri论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada Univ Ontario, Inst Technol, Fac Sci, 2000 Simcoe St North, Oshawa, ON L1H 7K4, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaPoda, Gennady论文数: 0 引用数: 0 h-index: 0机构: Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, Canada Univ Toronto, Leslie Dan Fac Pharm, 144 Coll St, Toronto, ON M5S 3M2, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaWu, Hong论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaDong, Aiping论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaKuznetsova, Ekaterina论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada React Biol Corp, Prod Dev, 1 Great Valley Pkwy,Suite 18, Malvern, PA 19355 USA Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaMarcellus, Richard论文数: 0 引用数: 0 h-index: 0机构: Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaSenisterra, Guillermo论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaDombrovski, Ludmila论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, Canada论文数: 引用数: h-index:机构:Kiyota, Taira论文数: 0 引用数: 0 h-index: 0机构: Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, Canada论文数: 引用数: h-index:机构:Arrowsmith, Cheryl H.论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaBrown, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaVedadi, Masoud论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, MaRS Ctr, 101 Coll St,South Tower, Toronto, ON M5G 1L7, Canada Univ Toronto, Dept Pharmacol & Toxicol, Med Sci Bldg,1 Kings Coll Circle, Toronto, ON M5S 1A8, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, CanadaAl-awar, Rima论文数: 0 引用数: 0 h-index: 0机构: Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, Canada Univ Toronto, Dept Pharmacol & Toxicol, Med Sci Bldg,1 Kings Coll Circle, Toronto, ON M5S 1A8, Canada Ontario Inst Canc Res, Drug Discovery Program, MaRS Ctr, 661 Univ Ave,West Tower, Toronto, ON M5G 0A3, Canada
- [10] Wdr5, a WD-40 protein, regulates osteoblast differentiation during embryonic bone developmentDEVELOPMENTAL BIOLOGY, 2006, 295 (02) : 498 - 506Gori, Francesca论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Massachusetts Gen Hosp, Endocrine Unit, Boston, MA 02114 USA Harvard Univ, Sch Med, Massachusetts Gen Hosp, Endocrine Unit, Boston, MA 02114 USAFriedman, Lauren G.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Massachusetts Gen Hosp, Endocrine Unit, Boston, MA 02114 USA Harvard Univ, Sch Med, Massachusetts Gen Hosp, Endocrine Unit, Boston, MA 02114 USADemay, Marie B.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Massachusetts Gen Hosp, Endocrine Unit, Boston, MA 02114 USA Harvard Univ, Sch Med, Massachusetts Gen Hosp, Endocrine Unit, Boston, MA 02114 USA