Synthesis and evaluation of salvinorin A analogues as kappa-opioid receptor ligands for the treatment of mood disorders.

被引：0
|
作者：
Beguin, C
Richards, MR
Liu-Chen, LY
Lee, DYW
Carlezon, WA
Cohen, BM
机构：
[1] Harvard Univ, Sch Med, McLean Hosp, Mol Pharmacol Lab, Belmont, MA 02478 USA
[2] Temple Univ, Sch Med, Dept Pharmacol, Philadelphia, PA 19122 USA
[3] McLean Hosp, HMS, Bioorgan & Nat Prod Lab, Belmont, MA 02178 USA
[4] McLean Hosp, HMS, Behav Genet Lab, Belmont, MA 02178 USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2005年 / 229卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
069-MEDI
引用
收藏
页码：U118 / U118
页数：1
相关论文
共 50 条
  • [1] Kappa-opioid ligands in the study and treatment of mood disorders
    Carlezon, William A., Jr.
    Beguin, Cecile
    Knoll, Allison T.
    Cohen, Bruce M.
    PHARMACOLOGY & THERAPEUTICS, 2009, 123 (03) : 334 - 343
  • [2] A review of salvinorin analogs and their kappa-opioid receptor activity
    Roach, Jeremy J.
    Shenvi, Ryan A.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 28 (09) : 1436 - 1445
  • [3] Kappa-opioid receptor ligands
    Husbands, SM
    EXPERT OPINION ON THERAPEUTIC PATENTS, 2004, 14 (12) : 1725 - 1741
  • [4] Kappa-opioid receptor-selective dicarboxylic ester-derived salvinorin A ligands
    Polepally, Prabhakar R.
    White, Kate
    Vardy, Eyal
    Roth, Bryan L.
    Ferreira, Daneel
    Zjawiony, Jordan K.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (10) : 2860 - 2862
  • [5] Syntheses of kappa-opioid receptor ligands: Salvinorin A analogs with modification at C-4 position.
    He, M
    Lee, DYW
    Liu-Chen, LY
    Ma, Z
    Wang, Y
    Chen, Y
    Carlezon, WA
    Beguin, C
    Cohen, BM
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 229 : U117 - U118
  • [6] Bioisosteric modification of salvinorin A, a potent and selective kappa-opioid receptor agonist
    Stewart, D. Jeremy
    Fahmy, Hesham
    Roth, Bryan L.
    Yan, Feng
    Zjawiony, Jordan K.
    ARZNEIMITTELFORSCHUNG-DRUG RESEARCH, 2006, 56 (04): : 269 - 275
  • [7] Synthesis of salvinorin A analogues as opioid receptor probes
    Tidgewell, Kevin
    Harding, Wayne W.
    Lozama, Anthony
    Cobb, Howard
    Shah, Kushal
    Kannan, Pavitra
    Dersch, Christina M.
    Parrish, Damon
    Deschamps, Jeffrey R.
    Rothman, Richard B.
    Prisinzano, Thomas E.
    JOURNAL OF NATURAL PRODUCTS, 2006, 69 (06): : 914 - 918
  • [8] Michael acceptor approach to the design of new salvinorin A-based high affinity ligands for the kappa-opioid receptor
    Polepally, Prabhakar R.
    Huben, Krzysztof
    Vardy, Eyal
    Setola, Vincent
    Mosier, Philip D.
    Roth, Bryan L.
    Zjawiony, Jordan K.
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 85 : 818 - 829
  • [9] SELECTIVE REVERSIBLE AND IRREVERSIBLE LIGANDS FOR THE KAPPA-OPIOID RECEPTOR
    CHENG, CY
    WU, SC
    HSIN, LW
    TAM, SW
    JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (12) : 2243 - 2247
  • [10] Models of neuroinflammation for the assessment of kappa-opioid receptor ligands
    Kalitin, K. Yu.
    Spasov, A. A.
    Mukha, O. Yu.
    PHARMACY & PHARMACOLOGY-FARMATSIYA I FARMAKOLOGIYA, 2023, 11 (01): : 4 - 18
12345